Design, synthesis and biological evaluation of novel 5-bromo derivatives of indole phytoalexins

  • Mariana Budovská,
  • Ivana Selešová,
  • Viera Tischlerová,
  • Radka Michalková and
  • Ján Mojžiš
Published 05 Mar 2020
Beilstein Arch. 2020, 202023. doi:10.3762/bxiv.2020.23.v1
Published 12 Feb 2020
Beilstein Arch. 2020, 202017. doi:10.3762/bxiv.2020.17.v1

Smart DNA biosensor for in vitro detection of androgen receptor mRNA

  • Ekaterina Alexandrovna Bryushkova,
  • Erik Rafikovich Gandalipov and
  • Julia Victorovna Nuzhina
Published 23 Jan 2020
Beilstein Arch. 2020, 202013. doi:10.3762/bxiv.2020.13.v1

Syntheses of xanthone derivatives and their bioactivity investigation

  • Beidou Zhou,
  • Zhimin Weng,
  • Yugui Tong,
  • Zetong Ma,
  • Rongrong Wei,
  • Jiali Li and
  • Zihan Yu
Published 27 Nov 2019
Beilstein Arch. 2019, 2019148. doi:10.3762/bxiv.2019.148.v1

NOVEL COMPOUNDS FROM CONDENSATION REACTION BETWEEN 2-ACETYLPYRIDINE AND 2-FORMYLPYRIDINE. SYNTHESIS, CRYSTAL STRUCTURE AND BIOLOGICAL EVALUATION

  • Roman Vasile Rusnac,
  • Maria Stefan Botnaru,
  • Nicanor Barba,
  • Peter Alexei Petrenko,
  • Yurii Chumakov and
  • Aurelian Petru Gulea
Published 18 Nov 2019
Beilstein Arch. 2019, 2019145. doi:10.3762/bxiv.2019.145.v1

Synthesis and cytotoxicity of novel oxindoles dispiro derivatives with thiohydantoin and adamantane fragments

  • Maxim E. Kukushkin,
  • Dmitriy A. Skvortsov,
  • Marina A. Kalinina,
  • Viktor A. Tafeenko,
  • Vladimir V. Burmistrov,
  • Gennady M. Butov,
  • Nikolai V. Zyk,
  • Alexander G. Majouga and
  • Elena K. Beloglazkina
Published 11 Nov 2019
Beilstein Arch. 2019, 2019143. doi:10.3762/bxiv.2019.143.v1
Published 17 Oct 2019
Beilstein Arch. 2019, 2019124. doi:10.3762/bxiv.2019.124.v1

Synthesis, structural characterization and biological activity of new pyrazolo[4,3-e][1,2,4]triazine acyclonucleosides

  • Mariusz Mojzych,
  • Zbigniew Karczmarzyk,
  • Joanna Matysiak and
  • Andrzej Fruziński
Published 09 Sep 2019
Beilstein Arch. 2019, 2019102. doi:10.3762/bxiv.2019.102.v1
Published 20 Aug 2019
Beilstein Arch. 2019, 201986. doi:10.3762/bxiv.2019.86.v1

An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agent

  • Nicky J Willis,
  • Elliott D Bayle,
  • George Papageorgiou,
  • David Steadman,
  • Benjamin N Aktinson,
  • William Mahy and
  • Paul V Fish
Published 16 Jul 2019
Beilstein Arch. 2019, 201970. doi:10.3762/bxiv.2019.70.v1

A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light

  • Xavier Gómez-Santacana,
  • Sabrina M. de Munnik,
  • Tamara A. M. Mocking,
  • Niels J. Hauwert,
  • Shanliang Sun,
  • Prashanna Vijayachandran,
  • Iwan J. P. de Esch,
  • Henry F. Vischer,
  • Maikel Wijtmans and
  • Rob Leurs
Published 15 Jul 2019
Beilstein Arch. 2019, 201969. doi:10.3762/bxiv.2019.69.v1

Azologization of a hetero-stilbene based c-RAF kinase inhibitor: Towards the design of photoswitchable sirtuin inhibitors

  • Christoph W. Grathwol,
  • Nathalie Wössner,
  • Sören Swyter,
  • Adam C. Smith,
  • Enrico Tapavicza,
  • Robert K. Hofstetter,
  • Anja Bodtke,
  • Manfred Jung and
  • Andreas Link
Published 01 Jul 2019
Beilstein Arch. 2019, 201953. doi:10.3762/bxiv.2019.53.v1

Characterization of two new degradation products of atorvastatin-calcium formed upon treatment with strong acids

  • Jürgen Krauß,
  • Monika Klimt,
  • Markus Luber,
  • Peter Mayer and
  • Franz Bracher
Published 28 May 2019
Beilstein Arch. 2019, 201931. doi:10.3762/bxiv.2019.31.v1
OTHER BEILSTEIN-INSTITUT OPEN SCIENCE ACTIVITIES