Design and Synthesis of Pyrene Containing Unusual α-Amino Acid Derivatives

  • Sambasivarao Kotha,
  • Vidyasagar Gaikwad and
  • Saima Ansari
Published 06 Oct 2022
Beilstein Arch. 2022, 202281. doi:10.3762/bxiv.2022.81.v1

Facile and Diastereoselective Arylation of the Privileged 1,4-Dihydroisoquinolin-3(2H)-one Scaffold

  • Dmitry Dar'in,
  • Grigory Kantin,
  • Alexander Bunev and
  • Mikhail Krasavin
Published 20 Jun 2022
Beilstein Arch. 2022, 202250. doi:10.3762/bxiv.2022.50.v1

Novel one-pot synthesis of 2-thio-substituted-3-H-phenothiazin-3-ones driven by oxidation with sodium periodate

  • Herman H. Odens Jr.,
  • Jae Y. You,
  • Alexandria D. Gallimore,
  • Preston H. Palm,
  • Cameron W. Davis,
  • Josue M. Bahena,
  • Jeffrey S. Moser,
  • Mackenzie E. Smith and
  • Herman H. Odens
Published 13 May 2022
Beilstein Arch. 2022, 202236. doi:10.3762/bxiv.2022.36.v1

New triazole triterpene derivative exhibits anti-RSV activity synthesis biological evaluation and molecular modeling

  • Elenilson Figueiredo da Silva,
  • Krist Helen Antunes Fernandes,
  • Denise Diedrich,
  • Jessica Gotardi,
  • Marcia Silvana Freire Franco,
  • Carlos Henrique Tomich de P da Silva,
  • Ana Paula Duarte de Souza and
  • Simone Cristina Baggio Gnoatto
Published 29 Apr 2022
Beilstein Arch. 2022, 202231. doi:10.3762/bxiv.2022.31.v1
Published 28 Feb 2022
Beilstein Arch. 2022, 202210. doi:10.3762/bxiv.2022.10.v1

The asymmetric Henry reaction as synthetic tool for production of drugs Linezolid and Rivaroxaban

  • Martin Vrbický,
  • Karel Macek,
  • Jaroslav Pochobradský,
  • Jan Svoboda,
  • Miloš Sedlák and
  • Pavel Drabina
Published 17 Jan 2022
Beilstein Arch. 2022, 20224. doi:10.3762/bxiv.2022.4.v1
Published 08 Nov 2021
Beilstein Arch. 2021, 202177. doi:10.3762/bxiv.2021.77.v1

First Total Synthesis of Hoshinoamides A  

  • Haipin Zhou,
  • Zihan Rui,
  • Yiming Yang,
  • Shengtao Xu,
  • Yutian Shao and
  • Long Liu
Published 15 Sep 2021
Beilstein Arch. 2021, 202164. doi:10.3762/bxiv.2021.64.v1

Host-guest interaction and properties of cucurbit[8]uril with chloramphenicol

  • Lin Zhang,
  • Jun Zheng,
  • Guangyan Luo,
  • Xiaoyue Li,
  • Yunqian Zhang,
  • Zhu Tao and
  • Qianjun Zhang
Published 30 Aug 2021
Beilstein Arch. 2021, 202162. doi:10.3762/bxiv.2021.62.v1

Ensemble-based virtual screening of Mycobacterium tuberculosis ClpC1 inhibitors

  • Hafsa Tayyab,
  • Nor F. W. Ridzwan and
  • Saharuddin B. Mohamad
Published 06 Jul 2021
Beilstein Arch. 2021, 202150. doi:10.3762/bxiv.2021.50.v1

Phenylamino pyrimidine-1,2,3-triazole derivatives as analogs of imatinib: searching for novel compounds against chronic myeloid leukemia

  • Luiz Claudio Ferreira Pimentel,
  • Lucas Villas Boas Hoelz,
  • Henayle Fernandes Canzian,
  • Frederico Silva Castelo Branco,
  • Andressa Paula de Oliveira,
  • Vinicius Rangel Campos,
  • Floriano Paes Silva Júnior,
  • Rafael Ferreira Dantas,
  • Jackson Antônio Lamounier Camargos Resende,
  • Anna Claudia Cunha,
  • Nubia Boechat and
  • Mônica Macedo Bastos
Published 09 Jun 2021
Beilstein Arch. 2021, 202144. doi:10.3762/bxiv.2021.44.v1

Design and synthesis of highly oxygenated furo[3,2-c]pyran-4-ones and furo[3,2-c]chromen-4-ones scaffold as potential anticancer and antimicrobial agent

  • Suman Rani,
  • Nisha Kamra,
  • Sumit Thakral,
  • Devinder Kumar,
  • Ajeet Singh,
  • Payare L Sangwan and
  • Shashank K Singh
Published 17 May 2021
Beilstein Arch. 2021, 202137. doi:10.3762/bxiv.2021.37.v1
Published 14 Apr 2021
Beilstein Arch. 2021, 202133. doi:10.3762/bxiv.2021.33.v1
Published 15 Mar 2021
Beilstein Arch. 2021, 202122. doi:10.3762/bxiv.2021.22.v1

Enhanced cell target specificity and uptake of lipid nanoparticles using RNA aptamers and peptides

  • Roslyn M. Ray,
  • Anders Højgaard Hansen,
  • Maria Taskova,
  • Bernhard Jandl,
  • Jonas Hansen,
  • Citra Soemardy,
  • Kevin V. Morris and
  • Kira Astakhova
Published 26 Jan 2021
Beilstein Arch. 2021, 20217. doi:10.3762/bxiv.2021.7.v1

Borylated methyl cinnamates: Expedited synthesis, characterization, crystallographic analysis and biological activities in glycosidase inhibition and in cancer cells lines.

  • William J Legge,
  • Yuna Shimadate,
  • Mahdi Ghorbani,
  • Jennette Sakoff,
  • Todd A Houston,
  • Atsushi Kato,
  • Paul Bernhardt and
  • Michela I. Simone
Published 22 Jan 2021
Beilstein Arch. 2021, 20214. doi:10.3762/bxiv.2021.4.v1

β-Lactamase inhibition profile of new amidine substituted diazabicyclooctanes

  • zafar iqbal,
  • Yuanyu Gao,
  • Dong Tang,
  • Xueqin Ma,
  • Jinbo Ji,
  • Jian Sun,
  • Jingwen Ji,
  • Yuanbai Liu,
  • Lijuan Zhai,
  • Rui Jiang,
  • Yangxiu Mu,
  • Lili He,
  • Haikang Yang and
  • Zhixiang Yang
Published 21 Dec 2020
Beilstein Arch. 2020, 2020143. doi:10.3762/bxiv.2020.143.v1
Published 08 Dec 2020
Beilstein Arch. 2020, 2020138. doi:10.3762/bxiv.2020.138.v1
Published 30 Nov 2020
Beilstein Arch. 2020, 2020135. doi:10.3762/bxiv.2020.135.v1
Published 26 Nov 2020
Beilstein Arch. 2020, 2020133. doi:10.3762/bxiv.2020.133.v1

Synthesis of 1-Indolyl-3,5,8-Substituted γ-Carbolines: One Pot Metal-Solvent Free Protocol and Biological Evaluation

  • Premansh Dudhe,
  • Mena Asha Krishnan,
  • Kratika Yadav,
  • Diptendu Roy,
  • Krishnan Venkatasubbaiah,
  • Biswarup Pathak and
  • Venkatesh Chelvam
Published 19 Nov 2020
Beilstein Arch. 2020, 2020131. doi:10.3762/bxiv.2020.131.v1

In silico approach: Anthocyanin derivatives as potential inhibitors of the COVID-19 main protease

  • Muhammad Ikhlas Abdjan,
  • Khusna Arif Rakhman,
  • Sri Handayani,
  • Chairil Anjasmara Robo Putra and
  • Imam Siswanto
Published 15 Sep 2020
Beilstein Arch. 2020, 2020106. doi:10.3762/bxiv.2020.106.v1

Vicinal difluorination as a C=C surrogate: an analog of piperine with enhanced solubility, photostability, and acetylcholinesterase inhibitory activity

  • Yuvixza Lizarme-Salas,
  • Alexandra Daryl Ariawan,
  • Ranjala Ratnayake,
  • Hendrik Luesch,
  • Angela Finch and
  • Luke Hunter
Published 12 Aug 2020
Beilstein Arch. 2020, 202093. doi:10.3762/bxiv.2020.93.v1
Published 08 May 2020
Beilstein Arch. 2020, 202060. doi:10.3762/bxiv.2020.60.v1
Published 27 Apr 2020
Beilstein Arch. 2020, 202055. doi:10.3762/bxiv.2020.55.v1
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