Factors governing the affinity and selectivity of histone deacetylase inhibitors for the HDAC8 enzyme active site: Implications for anticancer therapy

  1. Nikolay Toshev,
  2. Diana Cheshmedzhieva and
  3. Todor Dudev

Published 21 Oct 2020

Beilstein Arch. 2020, 2020121. doi:10.3762/bxiv.2020.121.v1

Regioselective chemo-enzymatic syntheses of ferulate conjugates as chromogenic substrates for feruloyl esterases

  1. Olga Gherbovet,
  2. Fernando Ferreira,
  3. Apolline Clément,
  4. Mélanie Ragon,
  5. Julien Durand,
  6. Sophie Bozonnet,
  7. Michael J. O'Donohue and
  8. Régis Fauré

Published 16 Sep 2020

Beilstein Arch. 2020, 2020107. doi:10.3762/bxiv.2020.107.v1

In silico approach: Anthocyanin derivatives as potential inhibitors of the COVID-19 main protease

  1. Muhammad Ikhlas Abdjan,
  2. Khusna Arif Rakhman,
  3. Sri Handayani,
  4. Chairil Anjasmara Robo Putra and
  5. Imam Siswanto

Published 15 Sep 2020

Beilstein Arch. 2020, 2020106. doi:10.3762/bxiv.2020.106.v1

Changed reactivity of secondary hydroxyl groups in C8-modified adenosine – lessons learned from silylation

  1. Jennifer Frommer and
  2. Sabine Müller

Published 09 Sep 2020

Beilstein Arch. 2020, 2020102. doi:10.3762/bxiv.2020.102.v1

Leveraging glycomics data in glycoprotein 3D structure validation with Privateer

  1. Haroldas Bagdonas,
  2. Daniel Ungar and
  3. Jon Agirre

Published 20 Jul 2020

Beilstein Arch. 2020, 202083. doi:10.3762/bxiv.2020.83.v1

Dibenzocyclooctadiene Lignans from Artemisia sieversiana and Their Nitric Oxide Inhibitory Effects

  1. Xu-Dong Zhou,
  2. Chao-Xi Chen,
  3. Xi-Kang Zheng,
  4. Li-Min Gong,
  5. Ke-Wu Zeng,
  6. Wei Wang and
  7. Peng-Fei Tu

Published 26 May 2020

Beilstein Arch. 2020, 202064. doi:10.3762/bxiv.2020.64.v1

A Novel Sustainable Method to Prepare Glutaric Acid from Glucose

  1. Lei Hao,
  2. Chao Jie Li,
  3. Lian Bo Zhao,
  4. Xi Xian Xie and
  5. Kui Lu

Published 19 May 2020

Beilstein Arch. 2020, 202062. doi:10.3762/bxiv.2020.62.v1

A study on the synthesis of β-amino acids: the first synthesis of a bicyclic hemiaminal (3,3-dimethyl-1-(2,4,5-trifluorophenyl) tetrahydro-3H,5H-oxazolo[3,4-c] [1,3] oxazin-5-one)

  1. Ozlem Gundogdu,
  2. Ertan Sahin and
  3. Yunus Kara

Published 21 Apr 2020

Beilstein Arch. 2020, 202053. doi:10.3762/bxiv.2020.53.v1

Menthyl esterification allows chiral resolution for synthesis of artificial glutamate analogs

  1. Kenji Morokuma,
  2. Shuntaro Tsukamoto,
  3. Kei Miyako,
  4. Ryuichi Sakai,
  5. Raku Irie and
  6. Masato Oikawa

Published 07 Apr 2020

Beilstein Arch. 2020, 202045. doi:10.3762/bxiv.2020.45.v1

Reaction of indoles with aromatic fluoromethyl ketones: An efficient synthesis of trifluoromethyl-indolyl-phenylethanols using K2CO3/nBu4PBr in water

  1. Thanigaimalai Pillaiyar,
  2. Masoud Sedaghati and
  3. Gregor Schnakenburg

Published 12 Feb 2020

Beilstein Arch. 2020, 202017. doi:10.3762/bxiv.2020.17.v1

Smart DNA biosensor for in vitro detection of androgen receptor mRNA

  1. Ekaterina Alexandrovna Bryushkova,
  2. Erik Rafikovich Gandalipov and
  3. Julia Victorovna Nuzhina

Published 23 Jan 2020

Beilstein Arch. 2020, 202013. doi:10.3762/bxiv.2020.13.v1

Identification of a novel binding mechanism of quinoline based molecules with lactate dehydrogenase of Plasmodium falciparum

  1. Rahul Singh,
  2. Vijay Bhardwaj and
  3. Rituraj Purohit

Published 06 Dec 2019

Beilstein Arch. 2019, 2019153. doi:10.3762/bxiv.2019.153.v1

Synthesis and herbicidal activity of aryloxyacetic acid derivatives as HPPD inhibitors

  1. Man-Man Wang,
  2. Hao Huang,
  3. Lei Shu,
  4. Jian-Min Liu,
  5. Jian-Qiu Zhang,
  6. Yi-Le Yan and
  7. Da-Yong Zhang

Published 28 Nov 2019

Beilstein Arch. 2019, 2019150. doi:10.3762/bxiv.2019.150.v1

Syntheses of xanthone derivatives and their bioactivity investigation

  1. Beidou Zhou,
  2. Zhimin Weng,
  3. Yugui Tong,
  4. Zetong Ma,
  5. Rongrong Wei,
  6. Jiali Li and
  7. Zihan Yu

Published 27 Nov 2019

Beilstein Arch. 2019, 2019148. doi:10.3762/bxiv.2019.148.v1

Synthesis and cytotoxicity of novel oxindoles dispiro derivatives with thiohydantoin and adamantane fragments

  1. Maxim E. Kukushkin,
  2. Dmitriy A. Skvortsov,
  3. Marina A. Kalinina,
  4. Viktor A. Tafeenko,
  5. Vladimir V. Burmistrov,
  6. Gennady M. Butov,
  7. Nikolai V. Zyk,
  8. Alexander G. Majouga and
  9. Elena K. Beloglazkina

Published 11 Nov 2019

Beilstein Arch. 2019, 2019143. doi:10.3762/bxiv.2019.143.v1

Model compound met the key structural and spectroscopic features of [FeFe]-hydrogenase active site

  1. Li Hai,
  2. Tianyong Zhang,
  3. Shuang Jiang,
  4. Xiaoyuan Ma,
  5. Di Wang and
  6. Bin Li

Published 30 Oct 2019

Beilstein Arch. 2019, 2019136. doi:10.3762/bxiv.2019.136.v1

Synthesis of C-glycosyl phosphonate derivatives of 4-amino-4-deoxy-α-L-arabinose

  1. Lukáš Kerner and
  2. Paul Kosma

Published 24 Oct 2019

Beilstein Arch. 2019, 2019129. doi:10.3762/bxiv.2019.129.v1

Understanding the Role of Active Site Residues in CotB2 Catalysis Using a Cluster Model

  1. Keren Raz,
  2. Ronja Driller,
  3. Thomas Brück,
  4. Bernhard Loll and
  5. Dan Thomas Major

Published 26 Sep 2019

Beilstein Arch. 2019, 2019108. doi:10.3762/bxiv.2019.108.v1

Synthesis, structural characterization and biological activity of new pyrazolo[4,3-e][1,2,4]triazine acyclonucleosides

  1. Mariusz Mojzych,
  2. Zbigniew Karczmarzyk,
  3. Joanna Matysiak and
  4. Andrzej Fruziński

Published 09 Sep 2019

Beilstein Arch. 2019, 2019102. doi:10.3762/bxiv.2019.102.v1

Skeletocutins M-Q, biologically active compounds from the fruiting bodies of the basidiomycete Skeletocutis sp. collected in Africa  

  1. Tian Cheng,
  2. Clara Chepkirui,
  3. Cony Decock,
  4. Josphat C. Matasyoh and
  5. Marc Stadler

Published 22 Jul 2019

Beilstein Arch. 2019, 201974. doi:10.3762/bxiv.2019.74.v1

An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agent

  1. Nicky J Willis,
  2. Elliott D Bayle,
  3. George Papageorgiou,
  4. David Steadman,
  5. Benjamin N Aktinson,
  6. William Mahy and
  7. Paul V Fish

Published 16 Jul 2019

Beilstein Arch. 2019, 201970. doi:10.3762/bxiv.2019.70.v1

A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light

  1. Xavier Gómez-Santacana,
  2. Sabrina M. de Munnik,
  3. Tamara A. M. Mocking,
  4. Niels J. Hauwert,
  5. Shanliang Sun,
  6. Prashanna Vijayachandran,
  7. Iwan J. P. de Esch,
  8. Henry F. Vischer,
  9. Maikel Wijtmans and
  10. Rob Leurs

Published 15 Jul 2019

Beilstein Arch. 2019, 201969. doi:10.3762/bxiv.2019.69.v1

Archangelolide: Sesquiterpene lactone with immunobiological potential from Laserpitium archangelica

  1. Silvie Rimpelová,
  2. Michal Jurášek,
  3. Lucie Peterková,
  4. Jiří Bejček,
  5. Vojtěch Spiwok,
  6. Miloš Majdl,
  7. Michal Jirásko,
  8. Miloš Buděšínský,
  9. Juraj Harmatha,
  10. Eva Kmoníčková,
  11. Pavel Drašar and
  12. Tomáš Ruml

Published 04 Jun 2019

Beilstein Arch. 2019, 201938. doi:10.3762/bxiv.2019.38.v1

Design, synthesis and biological evaluation of immunostimulating mannosylated desmuramyl peptides

  1. Rosana Ribić,
  2. Ranko Stojković,
  3. Lidija Milković,
  4. Mariastefania Antica,
  5. Marko Cigler and
  6. Srđanka Tomić

Published 16 Apr 2019

Beilstein Arch. 2019, 20198. doi:10.3762/bxiv.2019.8.v1

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