Me3Al mediated domino nucleophilic addition/intramolecular cyclisation of 2-(2-oxo-2-phenylethyl)benzonitriles with amines; A convenient approach for the synthesis of substituted 1-aminoisoquinolines

  1. Midhun Sai Krishna Adusumalli,
  2. Lakshmi Narayana Sharma Konidena,
  3. Hima Bindu Gandham,
  4. Krishnaiah Kumari,
  5. Krishna Reddy Valluru,
  6. Satya Kameswara Rao Nidasanametla,
  7. Venkateswara Rao Battula and
  8. Hari Krishna Namballa

Published 22 Mar 2021

Beilstein Arch. 2021, 202126. doi:10.3762/bxiv.2021.26.v1

Synthesis of bis-aryloxyfluoromethanes

  1. Carl Recsei and
  2. Yaniv Barda

Published 09 Mar 2021

Beilstein Arch. 2021, 202119. doi:10.3762/bxiv.2021.19.v1

Synthesis of multiply fluorinated N-acetyl-D-glucosamine and D-galactosamine analogs via the corresponding deoxyfluorinated glucosazide and galactosazide thiodonors

  1. Vojtěch Hamala,
  2. Lucie Červenková Šťastná,
  3. Martin Kurfiřt,
  4. Petra Cuřínová,
  5. Martin Dračínský and
  6. Jindřich Karban

Published 11 Feb 2021

Beilstein Arch. 2021, 202110. doi:10.3762/bxiv.2021.10.v1

β-Lactamase inhibition profile of new amidine substituted diazabicyclooctanes

  1. zafar iqbal,
  2. Yuanyu Gao,
  3. Dong Tang,
  4. Xueqin Ma,
  5. Jinbo Ji,
  6. Jian Sun,
  7. Jingwen Ji,
  8. Yuanbai Liu,
  9. Lijuan Zhai,
  10. Rui Jiang,
  11. Yangxiu Mu,
  12. Lili He,
  13. Haikang Yang and
  14. Zhixiang Yang

Published 21 Dec 2020

Beilstein Arch. 2020, 2020143. doi:10.3762/bxiv.2020.143.v1

Published 14 Dec 2020

Beilstein Arch. 2020, 2020142. doi:10.3762/bxiv.2020.142.v1

Mesoionic tetrazolium-5-aminides: Synthesis, Molecular and Crystal Structures, UV-Vis Spectra, and DFT Calculations

  1. Vladislav A. Budevich,
  2. Sergei V. Voitekhovich,
  3. Alexander V. Zuraev,
  4. Vadim E. Matulis,
  5. Vitaly E. Matulis,
  6. Alexander S. Lyakhov,
  7. Ludmila S. Ivashkevich and
  8. Oleg A. Ivashkevich

Published 22 Oct 2020

Beilstein Arch. 2020, 2020122. doi:10.3762/bxiv.2020.122.v1

Vicinal difluorination as a C=C surrogate: an analog of piperine with enhanced solubility, photostability, and acetylcholinesterase inhibitory activity

  1. Yuvixza Lizarme-Salas,
  2. Alexandra Daryl Ariawan,
  3. Ranjala Ratnayake,
  4. Hendrik Luesch,
  5. Angela Finch and
  6. Luke Hunter

Published 12 Aug 2020

Beilstein Arch. 2020, 202093. doi:10.3762/bxiv.2020.93.v1

Mechanism of Base-Catalyzed Halogen Dance Reactions and the Role of Bromo-Bridged Transition States

  1. Nader Sakhaee,
  2. Yousef Fazaeli,
  3. Esmail Doustkhah,
  4. Sahar Sakhaee,
  5. Ahmad Takallou and
  6. Akbar Mobaraki

Published 27 Jul 2020

Beilstein Arch. 2020, 202086. doi:10.3762/bxiv.2020.86.v1

Transformation of 2H-1,2,3-benzothiadiazine 1,1-dioxides variously substituted at the aromatic ring, via nucleophilic substitution and demethylation reactions

  1. Imre Gyűjtő,
  2. Márta Porcs-Makkay,
  3. Ernák Ferenc Várda,
  4. Gyöngyvér Pusztai,
  5. Gábor Tóth,
  6. Gyula Simig and
  7. Balázs Volk

Published 16 Jun 2020

Beilstein Arch. 2020, 202073. doi:10.3762/bxiv.2020.73.v1

Published 06 Apr 2020

Beilstein Arch. 2020, 202040. doi:10.3762/bxiv.2020.40.v1

Synthesis of new fluorescent molecules having an aggregation-induced emission property derived from 4-fluoroisoxazoles

  1. Kazuyuki Sato,
  2. Akira Kawasaki,
  3. Yukiko Karuo,
  4. Atsushi Tarui,
  5. Kentaro Kawai and
  6. Masaaki Omote

Published 27 Mar 2020

Beilstein Arch. 2020, 202034. doi:10.3762/bxiv.2020.34.v1

Development of fluorinated benzils and bisbenzils as room-temperature phosphorescent molecules

  1. Shigeyuki Yamada,
  2. Takuya Higashida,
  3. Yizhou Wang,
  4. Masato Morita,
  5. Takuya Hosokai,
  6. Kaveendra Maduwantha,
  7. Kaveenga Rasika Koswattage and
  8. Tsutomu Konno

Published 23 Mar 2020

Beilstein Arch. 2020, 202031. doi:10.3762/bxiv.2020.31.v1

Decarboxylative Bromination of Thiazole Core and Consecutive Cross-Coupling Reactions

  1. Emma Freiberger,
  2. Eric Täuscher,
  3. Uwe Ritter,
  4. Nadine Eckert and
  5. Helmar Görls

Published 13 Mar 2020

Beilstein Arch. 2020, 202027. doi:10.3762/bxiv.2020.27.v1

Published 17 Feb 2020

Beilstein Arch. 2020, 202020. doi:10.3762/bxiv.2020.20.v1

Synthesis of C70-fragment Buckybowls Having Alkoxy Substituents

  1. Yumi Yakiyama,
  2. Shota Hishikawa and
  3. Hidehiro Sakurai

Published 13 Feb 2020

Beilstein Arch. 2020, 202018. doi:10.3762/bxiv.2020.18.v1

Synthesis and Properties of Tetrathiafulvalenes Bearing 6-Aryl-1,4-dithiafulvenes

  1. Aya Yoshimura,
  2. Hitoshi Kimura,
  3. Kohei Kagawa,
  4. Mayuka Yoshioka,
  5. Toshiki Itou,
  6. Dhananjayan Vasu,
  7. Takashi Shirahata,
  8. Hideki Yorimitsu and
  9. Yohji Misaki

Published 12 Feb 2020

Beilstein Arch. 2020, 202016. doi:10.3762/bxiv.2020.16.v1

Synthesis and cytotoxicity of novel oxindoles dispiro derivatives with thiohydantoin and adamantane fragments

  1. Maxim E. Kukushkin,
  2. Dmitriy A. Skvortsov,
  3. Marina A. Kalinina,
  4. Viktor A. Tafeenko,
  5. Vladimir V. Burmistrov,
  6. Gennady M. Butov,
  7. Nikolai V. Zyk,
  8. Alexander G. Majouga and
  9. Elena K. Beloglazkina

Published 11 Nov 2019

Beilstein Arch. 2019, 2019143. doi:10.3762/bxiv.2019.143.v1

Efficient Method for Propargylation of Aldehydes Promoted by Allenyl Boron Compounds under Microwave Irradiation

  1. Jucleiton JR Freitas,
  2. Queila PSB Freitas,
  3. Silvia RCP Andrade,
  4. Juliano CR Freitas,
  5. Roberta A Oliveira and
  6. Paulo H Menezes

Published 01 Nov 2019

Beilstein Arch. 2019, 2019138. doi:10.3762/bxiv.2019.138.v1

Published 06 Sep 2019

Beilstein Arch. 2019, 2019100. doi:10.3762/bxiv.2019.100.v1

Published 02 Sep 2019

Beilstein Arch. 2019, 201995. doi:10.3762/bxiv.2019.95.v1

Friedel-Crafts approach to the one-pot synthesis of methoxy substituted thioxanthylium salts

  1. Kenta Tanaka,
  2. Yuta Tanaka,
  3. Mami Kishimoto,
  4. Yujiro Hoshino and
  5. Kiyoshi Honda

Published 21 Jun 2019

Beilstein Arch. 2019, 201941. doi:10.3762/bxiv.2019.41.v1

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