Models of Necessity

  1. Timothy Clark and
  2. Martin G Hicks

Published 19 Jun 2020

Beilstein Arch. 2020, 202077. doi:10.3762/bxiv.2020.77.v1

Transformation of 2H-1,2,3-benzothiadiazine 1,1-dioxides variously substituted at the aromatic ring, via nucleophilic substitution and demethylation reactions

  1. Imre Gyűjtő,
  2. Márta Porcs-Makkay,
  3. Ernák Ferenc Várda,
  4. Gyöngyvér Pusztai,
  5. Gábor Tóth,
  6. Gyula Simig and
  7. Balázs Volk

Published 16 Jun 2020

Beilstein Arch. 2020, 202073. doi:10.3762/bxiv.2020.73.v1

Metal-free synthesis of phosphinoylchroman-4-ones via phosphinoylation/cyclization cascade mediated by K2S2O8

  1. Qiang Liu,
  2. Weibang Lu,
  3. Guanqun Xie and
  4. Xiaoxia Wang

Published 10 Jun 2020

Beilstein Arch. 2020, 202071. doi:10.3762/bxiv.2020.71.v1

One-Pot and Metal-Free Synthesis of 3-Arylated 4-Nitrophenols via Polyfunctionalized Cyclohexanones from β-Nitrostyrenes

  1. Haruyasu Asahara,
  2. Minami Hiraishi and
  3. Nagatoshi Nishiwaki

Published 22 May 2020

Beilstein Arch. 2020, 202063. doi:10.3762/bxiv.2020.63.v1

A Novel Sustainable Method to Prepare Glutaric Acid from Glucose

  1. Lei Hao,
  2. Chao Jie Li,
  3. Lian Bo Zhao,
  4. Xi Xian Xie and
  5. Kui Lu

Published 19 May 2020

Beilstein Arch. 2020, 202062. doi:10.3762/bxiv.2020.62.v1

Convenient Synthesis and Biological Evaluation of Bis(indolyl)methane Alkaloid and Bis(aryl)alkanes Derivatives with Anti-cancer Properties  

  1. Liang Qi,
  2. Linxia Xiao and
  3. Rui Lin

Published 08 May 2020

Beilstein Arch. 2020, 202060. doi:10.3762/bxiv.2020.60.v1

DFT Mechanistic Study on the Reaction of Benzenesulfonyl Azides with Oxabicyclic Alkenes

  1. Daniel Aboagye Akuamoah,
  2. Richard Tia and
  3. Evans Adei

Published 05 May 2020

Beilstein Arch. 2020, 202057. doi:10.3762/bxiv.2020.57.v1

Tuneable access to indole, indolone and cinnoline derivatives from a common 1,4-diketone Michael acceptor

  1. Dalel El-Marrouki,
  2. Sabrina Touchet,
  3. Abderrahmen Abdelli,
  4. Hédi M'Rabet,
  5. Mohamed Lotfi Efrit and
  6. Philippe C. Gros

Published 27 Apr 2020

Beilstein Arch. 2020, 202056. doi:10.3762/bxiv.2020.56.v1

Facile Synthesis of 7-Alkyl-1,2,3,4-tetrahydro-[1,8]-naphthyridines as Arginine Mimetics Using a Horner–Wadsworth–Emmons Based Approach

  1. Rhys A Lippa,
  2. John A Murphy and
  3. Tim Barrett

Published 27 Apr 2020

Beilstein Arch. 2020, 202055. doi:10.3762/bxiv.2020.55.v1

A study on the synthesis of β-amino acids: the first synthesis of a bicyclic hemiaminal (3,3-dimethyl-1-(2,4,5-trifluorophenyl) tetrahydro-3H,5H-oxazolo[3,4-c] [1,3] oxazin-5-one)

  1. Ozlem Gundogdu,
  2. Ertan Sahin and
  3. Yunus Kara

Published 21 Apr 2020

Beilstein Arch. 2020, 202053. doi:10.3762/bxiv.2020.53.v1

Two-step continuous-flow synthesis of α-terpineol

  1. Beatriz L C de Carvalho,
  2. Anderson R Aguillon,
  3. Raquel A C Leão and
  4. Rodrigo Octavio M. A. de Souza

Published 06 Apr 2020

Beilstein Arch. 2020, 202041. doi:10.3762/bxiv.2020.41.v1

Disposable Cartridge Concept for On-Demand Synthesis of Turbo Grignards, Knochel-Hauser Amides and Magnesium Alkoxides

  1. Mateo Berton,
  2. Kevin Sheehan,
  3. Andrea Adamo and
  4. D. Tyler McQuade

Published 06 Apr 2020

Beilstein Arch. 2020, 202040. doi:10.3762/bxiv.2020.40.v1

Synthesis of new fluorescent molecules having an aggregation-induced emission property derived from 4-fluoroisoxazoles

  1. Kazuyuki Sato,
  2. Akira Kawasaki,
  3. Yukiko Karuo,
  4. Atsushi Tarui,
  5. Kentaro Kawai and
  6. Masaaki Omote

Published 27 Mar 2020

Beilstein Arch. 2020, 202034. doi:10.3762/bxiv.2020.34.v1

Synthesis of pyrrolidinedione-fused hexahydropyrrolo[2,1-a]isoquinolines via three-component [3+2] cycloaddition followed by one-pot N-allylation and intramolecular Heck reactions

  1. Xiaoming Ma,
  2. Suzhi Meng,
  3. Xiaofeng Zhang,
  4. Qiang Zhang,
  5. Shenghu Yan,
  6. Yue Zhang and
  7. Wei Zhang

Published 16 Mar 2020

Beilstein Arch. 2020, 202028. doi:10.3762/bxiv.2020.28.v1

Decarboxylative Bromination of Thiazole Core and Consecutive Cross-Coupling Reactions

  1. Emma Freiberger,
  2. Eric Täuscher,
  3. Uwe Ritter,
  4. Nadine Eckert and
  5. Helmar Görls

Published 13 Mar 2020

Beilstein Arch. 2020, 202027. doi:10.3762/bxiv.2020.27.v1

Design, synthesis and biological evaluation of novel 5-bromo derivatives of indole phytoalexins

  1. Mariana Budovská,
  2. Ivana Selešová,
  3. Viera Tischlerová,
  4. Radka Michalková and
  5. Ján Mojžiš

Published 05 Mar 2020

Beilstein Arch. 2020, 202023. doi:10.3762/bxiv.2020.23.v1

Synthesis of aryl 2-bromo-2-chloro-1,1-difluoroethyl ethers mediated by a reaction between phenols and halothane

  1. Yukiko Karuo,
  2. Ayaka Kametani,
  3. Atsushi Tarui,
  4. Kazuyuki Sato,
  5. Kentaro Kawai and
  6. Masaaki Omote

Published 19 Feb 2020

Beilstein Arch. 2020, 202021. doi:10.3762/bxiv.2020.21.v1

Asymmetric Synthesis of CF2-Aziridines Enabled by Combined Strong Brønsted Acid Catalysis

  1. Xing-Fa Tan,
  2. Fa-Guang Zhang and
  3. Jun-An Ma

Published 17 Feb 2020

Beilstein Arch. 2020, 202020. doi:10.3762/bxiv.2020.20.v1

Reaction of indoles with aromatic fluoromethyl ketones: An efficient synthesis of trifluoromethyl-indolyl-phenylethanols using K2CO3/nBu4PBr in water

  1. Thanigaimalai Pillaiyar,
  2. Masoud Sedaghati and
  3. Gregor Schnakenburg

Published 12 Feb 2020

Beilstein Arch. 2020, 202017. doi:10.3762/bxiv.2020.17.v1

Synthesis and Properties of Tetrathiafulvalenes Bearing 6-Aryl-1,4-dithiafulvenes

  1. Aya Yoshimura,
  2. Hitoshi Kimura,
  3. Kohei Kagawa,
  4. Mayuka Yoshioka,
  5. Toshiki Itou,
  6. Dhananjayan Vasu,
  7. Takashi Shirahata,
  8. Hideki Yorimitsu and
  9. Yohji Misaki

Published 12 Feb 2020

Beilstein Arch. 2020, 202016. doi:10.3762/bxiv.2020.16.v1

Preparation and in situ use of unstable N-alkyl a-diazo-g-butyrolactams in RhII-catalyzed X-H insertion reactions

  1. Maria Eremeyeva,
  2. Daniil Zhukovsky,
  3. Dmitry Dar'in and
  4. Mikhail Krasavin

Published 07 Feb 2020

Beilstein Arch. 2020, 202015. doi:10.3762/bxiv.2020.15.v1

Copper-Catalyzed Remote C–H Arylation of Polycyclic Aromatic Hydrocarbons (PAHs)

  1. Anping Luo,
  2. Min Zhang,
  3. Zhangyi Fu,
  4. Jingbo Lan,
  5. Di Wu and
  6. Jingsong You

Published 20 Jan 2020

Beilstein Arch. 2020, 202011. doi:10.3762/bxiv.2020.11.v1

Palladium-Catalyzed Regio- and Stereoselective Synthesis of Aryl and 3-Indolyl Substituted-4-Methylene- isoquinolin-1(2H)-ones.

  1. Valeria Nori,
  2. Antonio Arcadi,
  3. Armando Carlone,
  4. Fabio Marinelli and
  5. Marco Chiarini

Published 14 Jan 2020

Beilstein Arch. 2020, 20208. doi:10.3762/bxiv.2020.8.v1

A Green and Facile Method for the Synthesis of Substituted 1,2-Epoxy Ethylgembisphosphonates and their Symmetrical Dibutylammmonium Salts

  1. Siphamandla B. Simelane,
  2. Derek T. Ndinteh and
  3. Xavier Y. Mbianda

Published 06 Jan 2020

Beilstein Arch. 2020, 20203. doi:10.3762/bxiv.2020.3.v1

Straightforward convergent access to 2-arylated polysubstituted benzothiazoles

  1. Omar Sadek,
  2. David M Perrin and
  3. Emmanuel Gras

Published 05 Dec 2019

Beilstein Arch. 2019, 2019152. doi:10.3762/bxiv.2019.152.v1

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