An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agent

  1. Nicky J Willis,
  2. Elliott D Bayle,
  3. George Papageorgiou,
  4. David Steadman,
  5. Benjamin N Aktinson,
  6. William Mahy and
  7. Paul V Fish

Published 16 Jul 2019

Beilstein Arch. 2019, 201970. doi:10.3762/bxiv.2019.70.v1

Palladium-catalyzed Conia-ene Reaction of 1-alkynylindolin-3-ones: a strategy for the construction of Pyrrolo[1,2-a]indoles

  1. Yong-Qin Tang,
  2. Xing-Hai Fei,
  3. Jian-Xiong An,
  4. Fen-Fen Yang,
  5. Dong-Zhu Duan,
  6. Zuo-Xian Cao,
  7. Xiao-Zhong Fu,
  8. Yuan-Yong Yang,
  9. Bin He and
  10. Yong-Long Zhao

Published 04 Jul 2019

Beilstein Arch. 2019, 201959. doi:10.3762/bxiv.2019.59.v1

Synthesis of multi-substituted indene derivatives from aryl, vinyl, and alkyl/aryl carbinols

  1. Mithun Chakraborty,
  2. Gaddam Mahesh,
  3. Omkar R. Nakel,
  4. Gautamee Chavda,
  5. Susarla Anusha and
  6. Gangarajula Sudhakar

Published 07 Jun 2019

Beilstein Arch. 2019, 201939. doi:10.3762/bxiv.2019.39.v1

Synthesis of 1-azaspiro[4.4]nonan-1-oxyls via Intramolecular 1,3-Dipolar Cycloaddition

  1. Yulia V. Khoroshunova,
  2. Denis A. Morozov,
  3. Andrey I. Taratayko,
  4. Polina D. Gladkikh,
  5. Yuri I. Glazachev and
  6. Igor A. Kirilyuk

Published 03 Jun 2019

Beilstein Arch. 2019, 201937. doi:10.3762/bxiv.2019.37.v1

Installation of sulfonyl fluorides onto primary amides

  1. Jing Liu,
  2. Shi-Meng Wang and
  3. Hua-Li Qin

Published 29 May 2019

Beilstein Arch. 2019, 201933. doi:10.3762/bxiv.2019.33.v1

Characterization of two new degradation products of atorvastatin-calcium formed upon treatment with strong acids

  1. Jürgen Krauß,
  2. Monika Klimt,
  3. Markus Luber,
  4. Peter Mayer and
  5. Franz Bracher

Published 28 May 2019

Beilstein Arch. 2019, 201931. doi:10.3762/bxiv.2019.31.v1

Reaction of Arylmethyl Isocyanides/Arylmethyl-amines with Xanthate Esters: A Facile and Unexpected Synthesis of Carbamothioates

  1. Narasimhamurthy Rajeev,
  2. Toreshettahally R Swaroop,
  3. Seegehalli M Anil,
  4. Kupalli R Kiran,
  5. Chandru Chandru,
  6. Paris E Georghiou,
  7. Ahmad I Alrawashdeh,
  8. Shofiur Rahman,
  9. Abdullah Alodhayb,
  10. Kanchugarakoppal S Rangappa and
  11. Maralinganadoddi P Sadashiva

Published 21 May 2019

Beilstein Arch. 2019, 201926. doi:10.3762/bxiv.2019.26.v1

Published 23 Apr 2019

Beilstein Arch. 2019, 201914. doi:10.3762/bxiv.2019.14.v1

Application of Chiral 2-Isoxazoline for the Synthesis of syn-1,3-Diol Analogues

  1. Juanjuan Feng,
  2. Tianyu Li,
  3. Jiaxin Zhang and
  4. Peng Jiao

Published 17 Apr 2019

Beilstein Arch. 2019, 201910. doi:10.3762/bxiv.2019.10.v1

Reactions of 2-carbonyl and 2-hydroxy(or methoxy)alkyl substituted benzimidazoles with arenes in the superacid CF3SO3H. NMR and DFT study of dicationic electophilic species

  1. Dmitry Ryabukhin,
  2. Alexey Turdakov,
  3. Natalia Soldatova,
  4. Mikhail Kompanets,
  5. Alexander Ivanov,
  6. Irina Boyarskaya and
  7. Aleksander Vasilyev

Published 15 Apr 2019

Beilstein Arch. 2019, 20196. doi:10.3762/bxiv.2019.6.v1

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