Synthesis of new fluorescent molecules having an aggregation-induced emission property derived from 4-fluoroisoxazoles

  1. Kazuyuki Sato,
  2. Akira Kawasaki,
  3. Yukiko Karuo,
  4. Atsushi Tarui,
  5. Kentaro Kawai and
  6. Masaaki Omote

Published 27 Mar 2020

Beilstein Arch. 2020, 202034. doi:10.3762/bxiv.2020.34.v1

Synthesis of pyrrolidinedione-fused hexahydropyrrolo[2,1-a]isoquinolines via three-component [3+2] cycloaddition followed by one-pot N-allylation and intramolecular Heck reactions

  1. Xiaoming Ma,
  2. Suzhi Meng,
  3. Xiaofeng Zhang,
  4. Qiang Zhang,
  5. Shenghu Yan,
  6. Yue Zhang and
  7. Wei Zhang

Published 16 Mar 2020

Beilstein Arch. 2020, 202028. doi:10.3762/bxiv.2020.28.v1

Decarboxylative Bromination of Thiazole Core and Consecutive Cross-Coupling Reactions

  1. Emma Freiberger,
  2. Eric Täuscher,
  3. Uwe Ritter,
  4. Nadine Eckert and
  5. Helmar Görls

Published 13 Mar 2020

Beilstein Arch. 2020, 202027. doi:10.3762/bxiv.2020.27.v1

Design, synthesis and biological evaluation of novel 5-bromo derivatives of indole phytoalexins

  1. Mariana Budovská,
  2. Ivana Selešová,
  3. Viera Tischlerová,
  4. Radka Michalková and
  5. Ján Mojžiš

Published 05 Mar 2020

Beilstein Arch. 2020, 202023. doi:10.3762/bxiv.2020.23.v1

Synthesis of aryl 2-bromo-2-chloro-1,1-difluoroethyl ethers mediated by a reaction between phenols and halothane

  1. Yukiko Karuo,
  2. Ayaka Kametani,
  3. Atsushi Tarui,
  4. Kazuyuki Sato,
  5. Kentaro Kawai and
  6. Masaaki Omote

Published 19 Feb 2020

Beilstein Arch. 2020, 202021. doi:10.3762/bxiv.2020.21.v1

Asymmetric Synthesis of CF2-Aziridines Enabled by Combined Strong Brønsted Acid Catalysis

  1. Xing-Fa Tan,
  2. Fa-Guang Zhang and
  3. Jun-An Ma

Published 17 Feb 2020

Beilstein Arch. 2020, 202020. doi:10.3762/bxiv.2020.20.v1

Reaction of indoles with aromatic fluoromethyl ketones: An efficient synthesis of trifluoromethyl-indolyl-phenylethanols using K2CO3/nBu4PBr in water

  1. Thanigaimalai Pillaiyar,
  2. Masoud Sedaghati and
  3. Gregor Schnakenburg

Published 12 Feb 2020

Beilstein Arch. 2020, 202017. doi:10.3762/bxiv.2020.17.v1

Synthesis and Properties of Tetrathiafulvalenes Bearing 6-Aryl-1,4-dithiafulvenes

  1. Aya Yoshimura,
  2. Hitoshi Kimura,
  3. Kohei Kagawa,
  4. Mayuka Yoshioka,
  5. Toshiki Itou,
  6. Dhananjayan Vasu,
  7. Takashi Shirahata,
  8. Hideki Yorimitsu and
  9. Yohji Misaki

Published 12 Feb 2020

Beilstein Arch. 2020, 202016. doi:10.3762/bxiv.2020.16.v1

Preparation and in situ use of unstable N-alkyl a-diazo-g-butyrolactams in RhII-catalyzed X-H insertion reactions

  1. Maria Eremeyeva,
  2. Daniil Zhukovsky,
  3. Dmitry Dar'in and
  4. Mikhail Krasavin

Published 07 Feb 2020

Beilstein Arch. 2020, 202015. doi:10.3762/bxiv.2020.15.v1

Copper-Catalyzed Remote C–H Arylation of Polycyclic Aromatic Hydrocarbons (PAHs)

  1. Anping Luo,
  2. Min Zhang,
  3. Zhangyi Fu,
  4. Jingbo Lan,
  5. Di Wu and
  6. Jingsong You

Published 20 Jan 2020

Beilstein Arch. 2020, 202011. doi:10.3762/bxiv.2020.11.v1

Palladium-Catalyzed Regio- and Stereoselective Synthesis of Aryl and 3-Indolyl Substituted-4-Methylene- isoquinolin-1(2H)-ones.

  1. Valeria Nori,
  2. Antonio Arcadi,
  3. Armando Carlone,
  4. Fabio Marinelli and
  5. Marco Chiarini

Published 14 Jan 2020

Beilstein Arch. 2020, 20208. doi:10.3762/bxiv.2020.8.v1

A Green and Facile Method for the Synthesis of Substituted 1,2-Epoxy Ethylgembisphosphonates and their Symmetrical Dibutylammmonium Salts

  1. Siphamandla B. Simelane,
  2. Derek T. Ndinteh and
  3. Xavier Y. Mbianda

Published 06 Jan 2020

Beilstein Arch. 2020, 20203. doi:10.3762/bxiv.2020.3.v1

Straightforward convergent access to 2-arylated polysubstituted benzothiazoles

  1. Omar Sadek,
  2. David M Perrin and
  3. Emmanuel Gras

Published 05 Dec 2019

Beilstein Arch. 2019, 2019152. doi:10.3762/bxiv.2019.152.v1

Synthesis and herbicidal activity of aryloxyacetic acid derivatives as HPPD inhibitors

  1. Man-Man Wang,
  2. Hao Huang,
  3. Lei Shu,
  4. Jian-Min Liu,
  5. Jian-Qiu Zhang,
  6. Yi-Le Yan and
  7. Da-Yong Zhang

Published 28 Nov 2019

Beilstein Arch. 2019, 2019150. doi:10.3762/bxiv.2019.150.v1

Syntheses of xanthone derivatives and their bioactivity investigation

  1. Beidou Zhou,
  2. Zhimin Weng,
  3. Yugui Tong,
  4. Zetong Ma,
  5. Rongrong Wei,
  6. Jiali Li and
  7. Zihan Yu

Published 27 Nov 2019

Beilstein Arch. 2019, 2019148. doi:10.3762/bxiv.2019.148.v1

KOtBu Promoted Selective Ring-Opening N-alkylation of 2-Oxazolines to Access 2-Aminoethyl Acetates and N-Substituted Thiazolidinones

  1. Qiao Lin,
  2. Shiling Zhang and
  3. Bin Li

Published 19 Nov 2019

Beilstein Arch. 2019, 2019146. doi:10.3762/bxiv.2019.146.v1

NOVEL COMPOUNDS FROM CONDENSATION REACTION BETWEEN 2-ACETYLPYRIDINE AND 2-FORMYLPYRIDINE. SYNTHESIS, CRYSTAL STRUCTURE AND BIOLOGICAL EVALUATION

  1. Roman Vasile Rusnac,
  2. Maria Stefan Botnaru,
  3. Nicanor Barba,
  4. Peter Alexei Petrenko,
  5. Yurii Chumakov and
  6. Aurelian Petru Gulea

Published 18 Nov 2019

Beilstein Arch. 2019, 2019145. doi:10.3762/bxiv.2019.145.v1

Practical method to obtain α-acetoxyketones promoted by (diacetoxyiodo)benzene and acetic acid

  1. Osvaldo J Quintana-Romero,
  2. Jorge Camacho-Ruiz and
  3. Armando Ariza-Castolo

Published 13 Nov 2019

Beilstein Arch. 2019, 2019144. doi:10.3762/bxiv.2019.144.v1

Microwave-assisted Synthesis of 2-Substituted 4,5,6,7-Tetrahydro-1,3-thiazepines from 4-Aminobutanol

  1. María C. Mollo,
  2. Natalia B. Kilimciler,
  3. Juan A. Bisceglia and
  4. Liliana R. Orelli

Published 28 Oct 2019

Beilstein Arch. 2019, 2019135. doi:10.3762/bxiv.2019.135.v1

Straightforward Synthesis of Various Chiral Pyrimidines Bearing Stereogenic Center at the C2 position, Including C-Terminal Peptide Isosters

  1. Sami Sahtel,
  2. Rafâa Besbes,
  3. Emmanuel Vrancken and
  4. Jean-Marc Campagne

Published 28 Oct 2019

Beilstein Arch. 2019, 2019134. doi:10.3762/bxiv.2019.134.v1

Total synthesis of 2'-O-methyl-β-L-arabinosyluridine and reassignment the nucleoside from Penicillium sp. as 2'-O-methyl-β-L-uridine

  1. chunyang shen,
  2. Haixin Ding,
  3. Xueping Tao,
  4. Ruchun Yang,
  5. Jiang Bai,
  6. Banpeng Cao,
  7. Yiyuan Peng and
  8. Qiang Xiao

Published 23 Oct 2019

Beilstein Arch. 2019, 2019128. doi:10.3762/bxiv.2019.128.v1

Photosensitizer-Promoted Photoaddition Reactions of α-Silyl Group Containing N-Alkyl Glycinates to Dimethyl Acetylenedicarboxylate (DMAD)

  1. Suk Hyun Lim and
  2. Dae Won Cho

Published 15 Oct 2019

Beilstein Arch. 2019, 2019121. doi:10.3762/bxiv.2019.121.v1

Synthesis, structural characterization and biological activity of new pyrazolo[4,3-e][1,2,4]triazine acyclonucleosides

  1. Mariusz Mojzych,
  2. Zbigniew Karczmarzyk,
  3. Joanna Matysiak and
  4. Andrzej Fruziński

Published 09 Sep 2019

Beilstein Arch. 2019, 2019102. doi:10.3762/bxiv.2019.102.v1

Straightforward chemical desymmetrisation of cis-(±)-4-O-protected-cyclopent-2-enol using resolving agents on column chromatography

  1. Bemba Sidi Mohamed,
  2. Suzanne Peyrottes,
  3. Jean-Pierre Uttaro and
  4. Christophe MATHE

Published 03 Sep 2019

Beilstein Arch. 2019, 201998. doi:10.3762/bxiv.2019.98.v1

A Highly Efficient and Air-Insensitive Copper-Catalyzed Synthesis of Diorganyl Chalcogenides

  1. Yasamin Hamidian,
  2. Reza Mostafazadeh and
  3. Elmira Mohammadi

Published 28 Aug 2019

Beilstein Arch. 2019, 201992. doi:10.3762/bxiv.2019.92.v1

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