Cascade Intramolecular Prins/Friedel–Crafts Cyclization for the Synthesis of 4-Aryl-tetralin-2-ols and 5-Aryl-tetrahydro-5H-benzo[7]annulen-7-ols

  1. Jie Zheng,
  2. Shuyu Meng and
  3. Quan Rui Wang

Published 08 Mar 2021

Beilstein Arch. 2021, 202117. doi:10.3762/bxiv.2021.17.v1

Substituted Nitrogen-Bridged Diazocines

  1. Pascal Lentes,
  2. Jeremy Rudtke and
  3. Rainer Herges

Published 08 Mar 2021

Beilstein Arch. 2021, 202116. doi:10.3762/bxiv.2021.16.v1

Chiral Isothiourea-Catalyzed Kinetic Resolution of 4-Hydroxy[2.2]paracyclophane

  1. David Weinzierl and
  2. Mario Waser

Published 25 Feb 2021

Beilstein Arch. 2021, 202114. doi:10.3762/bxiv.2021.14.v1

Total Synthesis of Pyrrolo[2,3-c]quinoline Alkaloid: Trigonoine B

  1. Takashi Nishiyama,
  2. Erina Hamada,
  3. Daishi Ishii,
  4. Yuuto Kihara,
  5. Nanase Choshi,
  6. Natsumi Nakanishi,
  7. Mari Murakami,
  8. Kimiko Taninaka,
  9. Noriyuki Hatae and
  10. Tominari Choshi

Published 26 Jan 2021

Beilstein Arch. 2021, 20216. doi:10.3762/bxiv.2021.6.v1

Metal-free visible-light-enabled vicinal trifluoromethyl dithiolation of unactivated alkenes

  1. Xiaojuan Li,
  2. Qiang Zhang,
  3. Weigang Zhang,
  4. Jinzhu Ma,
  5. Yi Wang and
  6. Yi Pan

Published 13 Jan 2021

Beilstein Arch. 2021, 20211. doi:10.3762/bxiv.2021.1.v1

β-Lactamase inhibition profile of new amidine substituted diazabicyclooctanes

  1. zafar iqbal,
  2. Yuanyu Gao,
  3. Dong Tang,
  4. Xueqin Ma,
  5. Jinbo Ji,
  6. Jian Sun,
  7. Jingwen Ji,
  8. Yuanbai Liu,
  9. Lijuan Zhai,
  10. Rui Jiang,
  11. Yangxiu Mu,
  12. Lili He,
  13. Haikang Yang and
  14. Zhixiang Yang

Published 21 Dec 2020

Beilstein Arch. 2020, 2020143. doi:10.3762/bxiv.2020.143.v1

Synthesis of β-triazolylenones via metal-free desulfonylative alkylation of N-tosyl-1,2,3-triazoles

  1. Soumyaranjan Pati,
  2. Renata G. Almeida,
  3. Eufrânio N. da Silva Júnior and
  4. Irishi N. N. Namboothiri

Published 27 Nov 2020

Beilstein Arch. 2020, 2020134. doi:10.3762/bxiv.2020.134.v1

Synthesis of 1-Indolyl-3,5,8-Substituted γ-Carbolines: One Pot Metal-Solvent Free Protocol and Biological Evaluation

  1. Premansh Dudhe,
  2. Mena Asha Krishnan,
  3. Kratika Yadav,
  4. Diptendu Roy,
  5. Krishnan Venkatasubbaiah,
  6. Biswarup Pathak and
  7. Venkatesh Chelvam

Published 19 Nov 2020

Beilstein Arch. 2020, 2020131. doi:10.3762/bxiv.2020.131.v1

The Synthesis of Chiral β-Naphthyl-β-Sulfanyl Ketones via Enantioselective Sulfa-Michael Reaction in the Presence of a Bifunctional Cinchona/Sulfonamide Organocatalyst

  1. Deniz Tözendemir and
  2. Cihangir Tanyeli

Published 12 Nov 2020

Beilstein Arch. 2020, 2020129. doi:10.3762/bxiv.2020.129.v1

Synthesis of aminonaphthoquinone derivatives with Ceric Ammonium Nitrate (CAN) as a catalyst: NMR characterization and in silico reaction mechanism

  1. Jhoan H. Piermattey,
  2. Jhon Zapata-Rivera,
  3. Juan Oviedo,
  4. Ricardo Gaitan and
  5. Harold Gomez

Published 09 Nov 2020

Beilstein Arch. 2020, 2020128. doi:10.3762/bxiv.2020.128.v1

A Column-Free and Aqueous Waste-Free Process for Thioamide Preparation with Lawesson’s reagent

  1. Ke Wu,
  2. Yichen Ling,
  3. An Ding,
  4. Liqun Jin,
  5. Nan Sun,
  6. Baoxiang Hu,
  7. Zhenlu Shen and
  8. Xinquan Hu

Published 05 Nov 2020

Beilstein Arch. 2020, 2020126. doi:10.3762/bxiv.2020.126.v1

Au(III) Complexes with tetradentate cyclam based ligands

  1. Ann C Reiersølmoen,
  2. Thomas N Solvi and
  3. Anne Fiksdahl

Published 02 Nov 2020

Beilstein Arch. 2020, 2020124. doi:10.3762/bxiv.2020.124.v1

Facile Metal-Free Direct Transformation of N-Allyl- and tert-Butyl-Protected Arylamines to Azacycles Using Phosphoryl Chloride and TBD

  1. Van Hieu Tran,
  2. Wan Pyo Hong and
  3. Hee-Kwon Kim

Published 28 Oct 2020

Beilstein Arch. 2020, 2020123. doi:10.3762/bxiv.2020.123.v1

Mesoionic tetrazolium-5-aminides: Synthesis, Molecular and Crystal Structures, UV-Vis Spectra, and DFT Calculations

  1. Vladislav A. Budevich,
  2. Sergei V. Voitekhovich,
  3. Alexander V. Zuraev,
  4. Vadim E. Matulis,
  5. Vitaly E. Matulis,
  6. Alexander S. Lyakhov,
  7. Ludmila S. Ivashkevich and
  8. Oleg A. Ivashkevich

Published 22 Oct 2020

Beilstein Arch. 2020, 2020122. doi:10.3762/bxiv.2020.122.v1

Direct synthesis of anomeric tetrazolyl iminosugars from sugar-derived lactams

  1. Michał Mateusz Więcław and
  2. Bartłomiej Furman

Published 12 Oct 2020

Beilstein Arch. 2020, 2020118. doi:10.3762/bxiv.2020.118.v1

Metal-free synthesis of biarenes via photoextrusion in di(tri)arylphosphates

  1. Hisham Qrareya,
  2. Lorenzo Meazza,
  3. Stefano Protti and
  4. Maurizio Fagnoni

Published 28 Sep 2020

Beilstein Arch. 2020, 2020110. doi:10.3762/bxiv.2020.110.v1

Synthesis of 4-substituted azopyridine-functionalized Ni(II) porphyrins as molecular spin switches

  1. Jannis Ludwig,
  2. Tobias Moje,
  3. Fynn Röhricht and
  4. Rainer Herges

Published 25 Aug 2020

Beilstein Arch. 2020, 202096. doi:10.3762/bxiv.2020.96.v1

Three-Component Reactions of Aromatic Amines, 1,3-Dicarbonyl Compounds and α-Bromoacetaldehyde Acetal to Access N-Aryl/HetAryl-4,5-Unsubstituted Pyrroles

  1. Wenbo Huang,
  2. Kaimei Wang,
  3. Ping Liu,
  4. Shaoyong Ke and
  5. Yanlong Gu

Published 25 Aug 2020

Beilstein Arch. 2020, 202094. doi:10.3762/bxiv.2020.94.v1

A new method for the synthesis of diamantane by hydroisomerization of binor-S on treatment with sulfuric acid

  1. Rishat Aminov and
  2. Ravil I Khusnutdinov

Published 27 Jul 2020

Beilstein Arch. 2020, 202085. doi:10.3762/bxiv.2020.85.v1

Models of Necessity

  1. Timothy Clark and
  2. Martin G Hicks

Published 19 Jun 2020

Beilstein Arch. 2020, 202077. doi:10.3762/bxiv.2020.77.v1

Transformation of 2H-1,2,3-benzothiadiazine 1,1-dioxides variously substituted at the aromatic ring, via nucleophilic substitution and demethylation reactions

  1. Imre Gyűjtő,
  2. Márta Porcs-Makkay,
  3. Ernák Ferenc Várda,
  4. Gyöngyvér Pusztai,
  5. Gábor Tóth,
  6. Gyula Simig and
  7. Balázs Volk

Published 16 Jun 2020

Beilstein Arch. 2020, 202073. doi:10.3762/bxiv.2020.73.v1

Metal-free synthesis of phosphinoylchroman-4-ones via phosphinoylation/cyclization cascade mediated by K2S2O8

  1. Qiang Liu,
  2. Weibang Lu,
  3. Guanqun Xie and
  4. Xiaoxia Wang

Published 10 Jun 2020

Beilstein Arch. 2020, 202071. doi:10.3762/bxiv.2020.71.v1

One-Pot and Metal-Free Synthesis of 3-Arylated 4-Nitrophenols via Polyfunctionalized Cyclohexanones from β-Nitrostyrenes

  1. Haruyasu Asahara,
  2. Minami Hiraishi and
  3. Nagatoshi Nishiwaki

Published 22 May 2020

Beilstein Arch. 2020, 202063. doi:10.3762/bxiv.2020.63.v1

A Novel Sustainable Method to Prepare Glutaric Acid from Glucose

  1. Lei Hao,
  2. Chao Jie Li,
  3. Lian Bo Zhao,
  4. Xi Xian Xie and
  5. Kui Lu

Published 19 May 2020

Beilstein Arch. 2020, 202062. doi:10.3762/bxiv.2020.62.v1

Convenient Synthesis and Biological Evaluation of Bis(indolyl)methane Alkaloid and Bis(aryl)alkanes Derivatives with Anti-cancer Properties  

  1. Liang Qi,
  2. Linxia Xiao and
  3. Rui Lin

Published 08 May 2020

Beilstein Arch. 2020, 202060. doi:10.3762/bxiv.2020.60.v1

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