Synthesis, biological evaluation and molecular docking studies of new 2-ethoxy-4-{[3-alkyl(aryl)-4,5-dihydro-1H-1,2,4-triazol-5-on-4-yl]-azomethine}-phenyl benzenesulfonate derivatives on human aldose reductase enzyme

  1. Gül Özdemir,
  2. Namık Kılınç,
  3. Sevda Manap,
  4. Murat Beytur,
  5. Muzaffer Alkan and
  6. Haydar Yüksek

Published 06 Apr 2021

Beilstein Arch. 2021, 202131. doi:10.3762/bxiv.2021.31.v1

Organocatalytic Asymmetric Michael/Acyl Transfer Reaction between α-Nitroketones and 4-Arylidene- pyrrolidine-2,3-diones

  1. Chandrakanta Parida and
  2. Subhas C Pan

Published 23 Mar 2021

Beilstein Arch. 2021, 202128. doi:10.3762/bxiv.2021.28.v1

Me3Al mediated domino nucleophilic addition/intramolecular cyclisation of 2-(2-oxo-2-phenylethyl)benzonitriles with amines; A convenient approach for the synthesis of substituted 1-aminoisoquinolines

  1. Midhun Sai Krishna Adusumalli,
  2. Lakshmi Narayana Sharma Konidena,
  3. Hima Bindu Gandham,
  4. Krishnaiah Kumari,
  5. Krishna Reddy Valluru,
  6. Satya Kameswara Rao Nidasanametla,
  7. Venkateswara Rao Battula and
  8. Hari Krishna Namballa

Published 22 Mar 2021

Beilstein Arch. 2021, 202126. doi:10.3762/bxiv.2021.26.v1

Chemical synthesis of C6-tetrazole D-mannose building blocks and access to a bioisostere of mannuronic acid 1-phosphate

  1. Eleni Dimitriou and
  2. Gavin J Miller

Published 22 Mar 2021

Beilstein Arch. 2021, 202125. doi:10.3762/bxiv.2021.25.v1

Synthesis of polycyclic hydrocarbons C14H20 by hydrogenation of exo-exo-, exo-endo-, endo-exo-, and endo-endo- hexacyclo[9.2.1.02,10.03,8.04,6.05,9]tetradec-12-enes with H2SO4 and isomerization of the products to diamantane induced by ionic liquids

  1. Rishat Aminov and
  2. Ravil Khusnutdinov

Published 18 Mar 2021

Beilstein Arch. 2021, 202124. doi:10.3762/bxiv.2021.24.v1

Development of QSAR ensemble models for predicting the PAMPA Effective Permeability of new, non-peptidic leads with potential antiviral activity against the coronavirus SARS-CoV-2.

  1. Chrysoula Gousiadou,
  2. Philip Doganis and
  3. Haralambos Sarimveis

Published 15 Mar 2021

Beilstein Arch. 2021, 202122. doi:10.3762/bxiv.2021.22.v1

Structural Effects of meso-Halogenation on Porphyrins: meso-Xn-ABCD Macrocycles

  1. Keith J. Flanagan,
  2. Maximilian Paradiz Dominguez,
  3. Zoi Melissari,
  4. Hans-Georg Eckhardt,
  5. René M. Williams,
  6. Dáire Gibbons,
  7. Caroline Prior,
  8. Gemma M. Locke,
  9. Alina Meindl,
  10. Aoife A. Ryan and
  11. Mathias O Senge

Published 12 Mar 2021

Beilstein Arch. 2021, 202121. doi:10.3762/bxiv.2021.21.v1

Synthesis and transformation of sphingosine analogue pinane-based 2-amino-1,3-diols

  1. Ákos Bajtel,
  2. Mounir Raji,
  3. Matti Haukka,
  4. Ferenc Fülöp and
  5. Zsolt Szakonyi

Published 11 Mar 2021

Beilstein Arch. 2021, 202120. doi:10.3762/bxiv.2021.20.v1

Synthesis of bis-aryloxyfluoromethanes

  1. Carl Recsei and
  2. Yaniv Barda

Published 09 Mar 2021

Beilstein Arch. 2021, 202119. doi:10.3762/bxiv.2021.19.v1

DBU-catalyzed Michael addition of bulky glycine imine to α,β-unsaturated isoxazoles and pyrazolamides

  1. Yu-Jun Bai,
  2. Mei-Ling Cheng,
  3. Xiao-Mu Hu,
  4. Ya-Jun Bai,
  5. Xiao-Hui Zheng,
  6. Sheng-Yong Zhang and
  7. Ping-An Wang

Published 09 Mar 2021

Beilstein Arch. 2021, 202118. doi:10.3762/bxiv.2021.18.v1

Cascade Intramolecular Prins/Friedel–Crafts Cyclization for the Synthesis of 4-Aryl-tetralin-2-ols and 5-Aryl-tetrahydro-5H-benzo[7]annulen-7-ols

  1. Jie Zheng,
  2. Shuyu Meng and
  3. Quan Rui Wang

Published 08 Mar 2021

Beilstein Arch. 2021, 202117. doi:10.3762/bxiv.2021.17.v1

Substituted Nitrogen-Bridged Diazocines

  1. Pascal Lentes,
  2. Jeremy Rudtke and
  3. Rainer Herges

Published 08 Mar 2021

Beilstein Arch. 2021, 202116. doi:10.3762/bxiv.2021.16.v1

Blue Light induced Coupling of N-Hydroxysulphonamides: An efficient and green Approach to Access Symmetrical Thiosulfonates

  1. Arvind Kumar Pandey,
  2. Akhilesh Kumar,
  3. Narsingh Verma and
  4. Santosh Kumar Srivastava

Published 05 Mar 2021

Beilstein Arch. 2021, 202115. doi:10.3762/bxiv.2021.15.v1

Chiral Isothiourea-Catalyzed Kinetic Resolution of 4-Hydroxy[2.2]paracyclophane

  1. David Weinzierl and
  2. Mario Waser

Published 25 Feb 2021

Beilstein Arch. 2021, 202114. doi:10.3762/bxiv.2021.14.v1

Computational model predicts protein binding sites of a luminescent ligand equipped with guanidiniocarbonyl-pyrrole groups

  1. Neda Rafieiolhosseini,
  2. Matthias Killa,
  3. Niklas Tötsch,
  4. Jean-Noël Grad,
  5. Alexander Höing,
  6. Christian Ottmann,
  7. Shirley K. Knauer,
  8. Jens Voskuhl and
  9. Daniel Hoffmann

Published 19 Feb 2021

Beilstein Arch. 2021, 202111. doi:10.3762/bxiv.2021.11.v1

Synthesis of multiply fluorinated N-acetyl-D-glucosamine and D-galactosamine analogs via the corresponding deoxyfluorinated glucosazide and galactosazide thiodonors

  1. Vojtěch Hamala,
  2. Lucie Červenková Šťastná,
  3. Martin Kurfiřt,
  4. Petra Cuřínová,
  5. Martin Dračínský and
  6. Jindřich Karban

Published 11 Feb 2021

Beilstein Arch. 2021, 202110. doi:10.3762/bxiv.2021.10.v1

Enhanced cell target specificity and uptake of lipid nanoparticles using RNA aptamers and peptides

  1. Roslyn M. Ray,
  2. Anders Højgaard Hansen,
  3. Maria Taskova,
  4. Bernhard Jandl,
  5. Jonas Hansen,
  6. Citra Soemardy,
  7. Kevin V. Morris and
  8. Kira Astakhova

Published 26 Jan 2021

Beilstein Arch. 2021, 20217. doi:10.3762/bxiv.2021.7.v1

Total Synthesis of Pyrrolo[2,3-c]quinoline Alkaloid: Trigonoine B

  1. Takashi Nishiyama,
  2. Erina Hamada,
  3. Daishi Ishii,
  4. Yuuto Kihara,
  5. Nanase Choshi,
  6. Natsumi Nakanishi,
  7. Mari Murakami,
  8. Kimiko Taninaka,
  9. Noriyuki Hatae and
  10. Tominari Choshi

Published 26 Jan 2021

Beilstein Arch. 2021, 20216. doi:10.3762/bxiv.2021.6.v1

Borylated methyl cinnamates: Expedited synthesis, characterization, crystallographic analysis and biological activities in glycosidase inhibition and in cancer cells lines.

  1. William J Legge,
  2. Yuna Shimadate,
  3. Mahdi Ghorbani,
  4. Jennette Sakoff,
  5. Todd A Houston,
  6. Atsushi Kato,
  7. Paul Bernhardt and
  8. Michela I. Simone

Published 22 Jan 2021

Beilstein Arch. 2021, 20214. doi:10.3762/bxiv.2021.4.v1

Metal-free visible-light-enabled vicinal trifluoromethyl dithiolation of unactivated alkenes

  1. Xiaojuan Li,
  2. Qiang Zhang,
  3. Weigang Zhang,
  4. Jinzhu Ma,
  5. Yi Wang and
  6. Yi Pan

Published 13 Jan 2021

Beilstein Arch. 2021, 20211. doi:10.3762/bxiv.2021.1.v1

β-Lactamase inhibition profile of new amidine substituted diazabicyclooctanes

  1. zafar iqbal,
  2. Yuanyu Gao,
  3. Dong Tang,
  4. Xueqin Ma,
  5. Jinbo Ji,
  6. Jian Sun,
  7. Jingwen Ji,
  8. Yuanbai Liu,
  9. Lijuan Zhai,
  10. Rui Jiang,
  11. Yangxiu Mu,
  12. Lili He,
  13. Haikang Yang and
  14. Zhixiang Yang

Published 21 Dec 2020

Beilstein Arch. 2020, 2020143. doi:10.3762/bxiv.2020.143.v1

Stereoselective syntheses of 3-aminocyclooctanetriols and halocyclooctanetriols

  1. Emine Salamci and
  2. Yunus Zozik

Published 14 Dec 2020

Beilstein Arch. 2020, 2020142. doi:10.3762/bxiv.2020.142.v1

DNA with zwitterionic and negatively charged phosphate modifications: formation of DNA triplexes, duplexes and cell permeability studies

  1. Yongdong Su,
  2. Maitsetseg Bayarjargal,
  3. Tracy K Hale and
  4. Vyacheslav V Filichev

Published 08 Dec 2020

Beilstein Arch. 2020, 2020138. doi:10.3762/bxiv.2020.138.v1

Synthesis and characterization of β-carboline fatty alcohol hybrids as potential biological active and antioxidant molecules

  1. Venkateshwarlu Kontham,
  2. Bhavya Ippakayala and
  3. Devarapaga Madhu

Published 30 Nov 2020

Beilstein Arch. 2020, 2020135. doi:10.3762/bxiv.2020.135.v1

Synthesis of β-triazolylenones via metal-free desulfonylative alkylation of N-tosyl-1,2,3-triazoles

  1. Soumyaranjan Pati,
  2. Renata G. Almeida,
  3. Eufrânio N. da Silva Júnior and
  4. Irishi N. N. Namboothiri

Published 27 Nov 2020

Beilstein Arch. 2020, 2020134. doi:10.3762/bxiv.2020.134.v1

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