Synthesis of 1,4-azaphosphinine pyrimidine nucleosides and their evaluation as inhibitors of human cytidine deaminase and APOBEC3A

  • Maksim V Kvach,
  • Stefan Harjes,
  • Harikrishnan M Kurup,
  • Geoffrey B Jameson,
  • Elena Harjes and
  • Vyacheslav V Filichev
Published 08 Feb 2024
Beilstein Arch. 2024, 20249. doi:10.3762/bxiv.2024.9.v1

I2/H2O2 mediated synthesis and photophysical properties of imidazole-fused heterocycles via [4+1] cyclization approach

  • Haonan Li,
  • Chenping Gao,
  • Qingjie Liu,
  • Yanchun Guo,
  • Shuxia Cao and
  • Yufen Zhao
Published 07 Feb 2024
Beilstein Arch. 2024, 20248. doi:10.3762/bxiv.2024.8.v1

Innovative Synthesis of Drug-like Molecules Using Tetrazole as Core Building Blocks

  • Jingyao Li,
  • Ajay L. Chandgude,
  • Qiang Zheng and
  • Alexander Dömling
Published 05 Feb 2024
Beilstein Arch. 2024, 20247. doi:10.3762/bxiv.2024.7.v1

Monitoring carbohydrate 3D structure quality with the Privateer database

  • Jordan S Dialpuri,
  • Haroldas Bagdonas,
  • Lucy C Schofield,
  • Phuong Thao Pham,
  • Lou Holland and
  • Jon Agirre
Published 31 Jan 2024
Beilstein Arch. 2024, 20246. doi:10.3762/bxiv.2024.6.v1

Skeletal rearrangement in the 6,8-dioxabicyclo[3.2.1]octan-4-ol ring-system promoted by thionyl chloride or Appel conditions

  • Martyn Jevric,
  • Julian Klepp,
  • Johannes Puschnig,
  • Oscar Lamb,
  • Christopher J Sumby and
  • Ben W Greatrex
Published 30 Jan 2024
Beilstein Arch. 2024, 20245. doi:10.3762/bxiv.2024.5.v1
Published 18 Jan 2024
Beilstein Arch. 2024, 20242. doi:10.3762/bxiv.2024.2.v1

Bismuth(III) Triflate: An Economical and Environmentally Friendly Catalyst for the Nazarov Reaction

  • Manoel Trindade Rodrigues Jr.,
  • Aline Silva Barroso de Oliveira,
  • Ralph da Costa Gomes,
  • Amanda Soares Hirata,
  • Lucas A Zeoly,
  • Hugo Santos,
  • João Arantes,
  • Catarina Sofia Mateus Reis-Silva,
  • João Agostinho Machado-Neto,
  • Leticia Veras Costa-Lotufo and
  • Fernando Coelho
Published 03 Jan 2024
Beilstein Arch. 2024, 20241. doi:10.3762/bxiv.2024.1.v1

Confirmation of the Stereochemistry of Spiroviolene

  • Yao Kong,
  • Yuanning Liu,
  • Kaibiao Wang,
  • Tao Wang,
  • Chen Wang,
  • Ben Ai,
  • Hongli Jia,
  • Guohui Pan,
  • Min Yin and
  • Zhengren Xu
Published 28 Dec 2023
Beilstein Arch. 2023, 202368. doi:10.3762/bxiv.2023.68.v1
Published 28 Dec 2023
Beilstein Arch. 2023, 202367. doi:10.3762/bxiv.2023.67.v1

Enantioselective synthesis of β-aryl-γ-lactam derivatives via Heck-Matsuda desymmetrization of N-protected 2,5-dihydro-1-H-pyrroles

  • Arnaldo G. de Oliveira Junior,
  • Marti F Wang,
  • Rafaela C Carmona,
  • Danilo M Lustosa,
  • Sergei A Gorbatov and
  • Carlos Roque D Correia
Published 28 Dec 2023
Beilstein Arch. 2023, 202366. doi:10.3762/bxiv.2023.66.v1

Spatial Arrangements of Cyclodextrin Host-Guest Complexes in Solution Studied by 13C-NMR and Molecular Modelling

  • Konstantin Lebedinskiy,
  • Ivan Barvík,
  • Zdeněk Tošner,
  • Ivana Císařová,
  • Jindřich Jindřich and
  • Radim Hrdina
Published 21 Dec 2023
Beilstein Arch. 2023, 202364. doi:10.3762/bxiv.2023.64.v1

Enzymatic evidence that the natural product N-nitroglycine is degraded by diverse bacteria

  • Kara A Strickland,
  • Brenda Martinez Rodriguez,
  • Ashley A Holland,
  • Shelby Wagner,
  • Michelle Luna-Alva,
  • David E Graham and
  • Jonathan D Caranto
Published 19 Dec 2023
Beilstein Arch. 2023, 202363. doi:10.3762/bxiv.2023.63.v1
Published 15 Dec 2023
Beilstein Arch. 2023, 202362. doi:10.3762/bxiv.2023.62.v1

Evaluation of the enantioselectivity of new chiral ligands based on imidazolidine-4-one derivatives

  • Jan Bartáček,
  • Karel Chlumský,
  • Jan Mrkvička,
  • Lucie Paloušová,
  • Miloš Sedlák and
  • Pavel Drabina
Published 14 Dec 2023
Beilstein Arch. 2023, 202361. doi:10.3762/bxiv.2023.61.v1
Published 13 Dec 2023
Beilstein Arch. 2023, 202360. doi:10.3762/bxiv.2023.60.v1
Published 11 Dec 2023
Beilstein Arch. 2023, 202359. doi:10.3762/bxiv.2023.59.v1

Chemical and Biosynthetic Potential of Penicillium shentong XL-F41

  • Ran Zou,
  • Xin Li,
  • Xiaochen Chen,
  • Yue-Wei Guo and
  • Baofu Xu
Published 07 Dec 2023
Beilstein Arch. 2023, 202358. doi:10.3762/bxiv.2023.58.v1

Nucleophilic Functionalization of Thianthrenium Salts under Base Conditions

  • Xinting Fan,
  • Duo Zhang,
  • xiangchuan xiu,
  • Bin Xu,
  • Yu Yuan,
  • Feng Chen and
  • Pan Gao
Published 07 Dec 2023
Beilstein Arch. 2023, 202357. doi:10.3762/bxiv.2023.57.v1

Genome Mining Reveals the Structure of the Clostrisin and Cellulosin Biosynthetic Gene Clusters, Two Novel Lantibiotics

  • Moisés Alejandro Alejo Hernandez,
  • Katia Pamela Villavicencio Sánchez,
  • Rosendo Sánchez Morales,
  • Karla Georgina Hernández-Magro Gil,
  • David Silverio Moreno-Gutiérrez,
  • Eddie Guillermo Sanchez-Rueda,
  • Yanet Teresa-Cruz,
  • Armando Hernández Garcia,
  • Alba Romero-Rodríguez,
  • Oscar Juárez,
  • Siseth Martínez-Caballero,
  • Mario Figueroa and
  • Corina Diana Ceapa
Published 06 Dec 2023
Beilstein Arch. 2023, 202356. doi:10.3762/bxiv.2023.56.v1
Published 05 Dec 2023
Beilstein Arch. 2023, 202355. doi:10.3762/bxiv.2023.55.v1
Published 28 Nov 2023
Beilstein Arch. 2023, 202354. doi:10.3762/bxiv.2023.54.v1

Facile Approach to the N,O,S-Heteropentacycles via Condensation of Sterically Crowded 3H-Phenoxazin-3-one with ortho-amino-, hydroxy- and mercaptoanilines

  • Eugeny P. Ivakhnenko,
  • Vasily I. Malay,
  • Pavel A. Knyazev,
  • Nikita I. Merezhko,
  • Nadezhda I. Makarova,
  • Oleg P. Demidov,
  • Gennady S. Borodkin,
  • Andrey G. Starikov and
  • Vladimir I. Minkin
Published 27 Nov 2023
Beilstein Arch. 2023, 202353. doi:10.3762/bxiv.2023.53.v1
Published 24 Nov 2023
Beilstein Arch. 2023, 202352. doi:10.3762/bxiv.2023.52.v1
Published 22 Nov 2023
Beilstein Arch. 2023, 202351. doi:10.3762/bxiv.2023.51.v1
Published 21 Nov 2023
Beilstein Arch. 2023, 202350. doi:10.3762/bxiv.2023.50.v1
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