Published 16 Jul 2019

Beilstein Arch. 2019, 201971. doi:10.3762/bxiv.2019.71.v1

An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agent

  1. Nicky J Willis,
  2. Elliott D Bayle,
  3. George Papageorgiou,
  4. David Steadman,
  5. Benjamin N Aktinson,
  6. William Mahy and
  7. Paul V Fish

Published 16 Jul 2019

Beilstein Arch. 2019, 201970. doi:10.3762/bxiv.2019.70.v1

A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light

  1. Xavier Gómez-Santacana,
  2. Sabrina M. de Munnik,
  3. Tamara A. M. Mocking,
  4. Niels J. Hauwert,
  5. Shanliang Sun,
  6. Prashanna Vijayachandran,
  7. Iwan J. P. de Esch,
  8. Henry F. Vischer,
  9. Maikel Wijtmans and
  10. Rob Leurs

Published 15 Jul 2019

Beilstein Arch. 2019, 201969. doi:10.3762/bxiv.2019.69.v1

Photochromic diarylethene with turn-off fluorescent switching property

  1. Luna Kono,
  2. Yuma Nakagawa,
  3. Ayako Fujimoto,
  4. Ryo Nishimura,
  5. Yohei Hattori,
  6. Toshiki Mutai,
  7. Nobuhiro Yasuda,
  8. Kenichi Koizumi,
  9. Satoshi Yokojima,
  10. Shinichiro Nakamura and
  11. Kingo Uchida

Published 11 Jul 2019

Beilstein Arch. 2019, 201966. doi:10.3762/bxiv.2019.66.v1

Synthesis of diastereomeric pheromones: adjacent methyl-branched alcohols and ketones

  1. VAN-DUNG LE,
  2. Chi-Hien Dang,
  3. Cong-Hao Nguyen,
  4. Van-Su Dang and
  5. Thanh-Danh Nguyen

Published 09 Jul 2019

Beilstein Arch. 2019, 201964. doi:10.3762/bxiv.2019.64.v1

1,3-Dipolar Cycloadditions of Isatin N,N′‑Cyclic Azomethine Imines with Alkynes for the synthesis of spiro[indoline-3,1'-pyrazolo[1,2-a]pyrazoles]

  1. Yang Shi,
  2. Gangqiang Wang,
  3. Zhiyu Chen,
  4. Minghu Wu,
  5. Jian Wang,
  6. Leslie Trigoura,
  7. Haibing Guo,
  8. Yalan Xing and
  9. Shaofa Sun

Published 08 Jul 2019

Beilstein Arch. 2019, 201963. doi:10.3762/bxiv.2019.63.v1

Palladium-catalyzed Conia-ene Reaction of 1-alkynylindolin-3-ones: a strategy for the construction of Pyrrolo[1,2-a]indoles

  1. Yong-Qin Tang,
  2. Xing-Hai Fei,
  3. Jian-Xiong An,
  4. Fen-Fen Yang,
  5. Dong-Zhu Duan,
  6. Zuo-Xian Cao,
  7. Xiao-Zhong Fu,
  8. Yuan-Yong Yang,
  9. Bin He and
  10. Yong-Long Zhao

Published 04 Jul 2019

Beilstein Arch. 2019, 201959. doi:10.3762/bxiv.2019.59.v1

Azologization of a hetero-stilbene based c-RAF kinase inhibitor: Towards the design of photoswitchable sirtuin inhibitors

  1. Christoph W. Grathwol,
  2. Nathalie Wössner,
  3. Sören Swyter,
  4. Adam C. Smith,
  5. Enrico Tapavicza,
  6. Robert K. Hofstetter,
  7. Anja Bodtke,
  8. Manfred Jung and
  9. Andreas Link

Published 01 Jul 2019

Beilstein Arch. 2019, 201953. doi:10.3762/bxiv.2019.53.v1

Sugar Derived Oxazolone Pseudotetrapeptide as γ-Turn Inducer and Anion-Selective Transporter

  1. Sachin S. Burade,
  2. Sushil V. Pawar,
  3. Tanmoy Saha,
  4. Navnath M Kumbhar,
  5. Amol S. Kotmale,
  6. Manzoor Ahmad,
  7. Pinaki Talukdar and
  8. Dilip D Dhavale

Published 27 Jun 2019

Beilstein Arch. 2019, 201949. doi:10.3762/bxiv.2019.49.v1

Ultrafast processes triggered by one- and two-photon excitation of a photochromic and luminescent hydrazone

  1. Alessandro Iagatti,
  2. Baihao Shao,
  3. Alberto Credi,
  4. Barbara Ventura,
  5. Ivan Aprahamian and
  6. Mariangela Di Donato

Published 27 Jun 2019

Beilstein Arch. 2019, 201948. doi:10.3762/bxiv.2019.48.v1

Excited State Dynamics for Visible Light Sensitization of Fast Photochromic Phenoxyl-Imidazolyl Radical Complex with Aryl Ketone

  1. Yoichi Kobayashi,
  2. Yukie Mamiya,
  3. Katsuya Mutoh,
  4. Hikaru Sotome,
  5. Masafumi Koga,
  6. Hiroshi Miyasaka and
  7. Jiro Abe

Published 24 Jun 2019

Beilstein Arch. 2019, 201946. doi:10.3762/bxiv.2019.46.v1

Friedel-Crafts approach to the one-pot synthesis of methoxy substituted thioxanthylium salts

  1. Kenta Tanaka,
  2. Yuta Tanaka,
  3. Mami Kishimoto,
  4. Yujiro Hoshino and
  5. Kiyoshi Honda

Published 21 Jun 2019

Beilstein Arch. 2019, 201941. doi:10.3762/bxiv.2019.41.v1

Synthesis of multi-substituted indene derivatives from aryl, vinyl, and alkyl/aryl carbinols

  1. Mithun Chakraborty,
  2. Gaddam Mahesh,
  3. Omkar R. Nakel,
  4. Gautamee Chavda,
  5. Susarla Anusha and
  6. Gangarajula Sudhakar

Published 07 Jun 2019

Beilstein Arch. 2019, 201939. doi:10.3762/bxiv.2019.39.v1

Archangelolide: Sesquiterpene lactone with immunobiological potential from Laserpitium archangelica

  1. Silvie Rimpelová,
  2. Michal Jurášek,
  3. Lucie Peterková,
  4. Jiří Bejček,
  5. Vojtěch Spiwok,
  6. Miloš Majdl,
  7. Michal Jirásko,
  8. Miloš Buděšínský,
  9. Juraj Harmatha,
  10. Eva Kmoníčková,
  11. Pavel Drašar and
  12. Tomáš Ruml

Published 04 Jun 2019

Beilstein Arch. 2019, 201938. doi:10.3762/bxiv.2019.38.v1

Synthesis of 1-azaspiro[4.4]nonan-1-oxyls via Intramolecular 1,3-Dipolar Cycloaddition

  1. Yulia V. Khoroshunova,
  2. Denis A. Morozov,
  3. Andrey I. Taratayko,
  4. Polina D. Gladkikh,
  5. Yuri I. Glazachev and
  6. Igor A. Kirilyuk

Published 03 Jun 2019

Beilstein Arch. 2019, 201937. doi:10.3762/bxiv.2019.37.v1

Installation of sulfonyl fluorides onto primary amides

  1. Jing Liu,
  2. Shi-Meng Wang and
  3. Hua-Li Qin

Published 29 May 2019

Beilstein Arch. 2019, 201933. doi:10.3762/bxiv.2019.33.v1

Characterization of two new degradation products of atorvastatin-calcium formed upon treatment with strong acids

  1. Jürgen Krauß,
  2. Monika Klimt,
  3. Markus Luber,
  4. Peter Mayer and
  5. Franz Bracher

Published 28 May 2019

Beilstein Arch. 2019, 201931. doi:10.3762/bxiv.2019.31.v1

Effect of Ring Size on Photoisomerization Properties of Stiff Stilbene macrocycles

  1. Sandra Olsson,
  2. Óscar Benito Pérez,
  3. Magnus Blom and
  4. Adolf Gogoll

Published 28 May 2019

Beilstein Arch. 2019, 201930. doi:10.3762/bxiv.2019.30.v1

Reaction of Arylmethyl Isocyanides/Arylmethyl-amines with Xanthate Esters: A Facile and Unexpected Synthesis of Carbamothioates

  1. Narasimhamurthy Rajeev,
  2. Toreshettahally R Swaroop,
  3. Seegehalli M Anil,
  4. Kupalli R Kiran,
  5. Chandru Chandru,
  6. Paris E Georghiou,
  7. Ahmad I Alrawashdeh,
  8. Shofiur Rahman,
  9. Abdullah Alodhayb,
  10. Kanchugarakoppal S Rangappa and
  11. Maralinganadoddi P Sadashiva

Published 21 May 2019

Beilstein Arch. 2019, 201926. doi:10.3762/bxiv.2019.26.v1

Tautomerism as primary signalling mechanism in metal sensing: the case of amide group

  1. Vera V. Deneva,
  2. Georgi Dobrikov,
  3. Aurelien Crochet,
  4. Daniela Nedeltcheva,
  5. Katharina M. Fromm and
  6. Liudmil Antonov

Published 20 May 2019

Beilstein Arch. 2019, 201923. doi:10.3762/bxiv.2019.23.v1

Published 14 May 2019

Beilstein Arch. 2019, 201922. doi:10.3762/bxiv.2019.22.v1

Published 07 May 2019

Beilstein Arch. 2019, 201919. doi:10.3762/bxiv.2019.19.v1

Published 23 Apr 2019

Beilstein Arch. 2019, 201914. doi:10.3762/bxiv.2019.14.v1

Diazocine functionalized TATA Platforms

  1. Roland Löw,
  2. Talina Rusch,
  3. Fynn Röhricht,
  4. Olaf M. Magnussen and
  5. Rainer Herges

Published 18 Apr 2019

Beilstein Arch. 2019, 201911. doi:10.3762/bxiv.2019.11.v1

Application of Chiral 2-Isoxazoline for the Synthesis of syn-1,3-Diol Analogues

  1. Juanjuan Feng,
  2. Tianyu Li,
  3. Jiaxin Zhang and
  4. Peng Jiao

Published 17 Apr 2019

Beilstein Arch. 2019, 201910. doi:10.3762/bxiv.2019.10.v1

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