Me3Al mediated domino nucleophilic addition/intramolecular cyclisation of 2-(2-oxo-2-phenylethyl)benzonitriles with amines; A convenient approach for the synthesis of substituted 1-aminoisoquinolines

  1. Midhun Sai Krishna Adusumalli,
  2. Lakshmi Narayana Sharma Konidena,
  3. Hima Bindu Gandham,
  4. Krishnaiah Kumari,
  5. Krishna Reddy Valluru,
  6. Satya Kameswara Rao Nidasanametla,
  7. Venkateswara Rao Battula and
  8. Hari Krishna Namballa

Published 22 Mar 2021

Beilstein Arch. 2021, 202126. doi:10.3762/bxiv.2021.26.v1

Published 15 Mar 2021

Beilstein Arch. 2021, 202122. doi:10.3762/bxiv.2021.22.v1

Enhanced cell target specificity and uptake of lipid nanoparticles using RNA aptamers and peptides

  1. Roslyn M. Ray,
  2. Anders Højgaard Hansen,
  3. Maria Taskova,
  4. Bernhard Jandl,
  5. Jonas Hansen,
  6. Citra Soemardy,
  7. Kevin V. Morris and
  8. Kira Astakhova

Published 26 Jan 2021

Beilstein Arch. 2021, 20217. doi:10.3762/bxiv.2021.7.v1

Borylated methyl cinnamates: Expedited synthesis, characterization, crystallographic analysis and biological activities in glycosidase inhibition and in cancer cells lines.

  1. William J Legge,
  2. Yuna Shimadate,
  3. Mahdi Ghorbani,
  4. Jennette Sakoff,
  5. Todd A Houston,
  6. Atsushi Kato,
  7. Paul Bernhardt and
  8. Michela I. Simone

Published 22 Jan 2021

Beilstein Arch. 2021, 20214. doi:10.3762/bxiv.2021.4.v1

β-Lactamase inhibition profile of new amidine substituted diazabicyclooctanes

  1. zafar iqbal,
  2. Yuanyu Gao,
  3. Dong Tang,
  4. Xueqin Ma,
  5. Jinbo Ji,
  6. Jian Sun,
  7. Jingwen Ji,
  8. Yuanbai Liu,
  9. Lijuan Zhai,
  10. Rui Jiang,
  11. Yangxiu Mu,
  12. Lili He,
  13. Haikang Yang and
  14. Zhixiang Yang

Published 21 Dec 2020

Beilstein Arch. 2020, 2020143. doi:10.3762/bxiv.2020.143.v1

Published 08 Dec 2020

Beilstein Arch. 2020, 2020138. doi:10.3762/bxiv.2020.138.v1

Published 30 Nov 2020

Beilstein Arch. 2020, 2020135. doi:10.3762/bxiv.2020.135.v1

Published 26 Nov 2020

Beilstein Arch. 2020, 2020133. doi:10.3762/bxiv.2020.133.v1

Synthesis of 1-Indolyl-3,5,8-Substituted γ-Carbolines: One Pot Metal-Solvent Free Protocol and Biological Evaluation

  1. Premansh Dudhe,
  2. Mena Asha Krishnan,
  3. Kratika Yadav,
  4. Diptendu Roy,
  5. Krishnan Venkatasubbaiah,
  6. Biswarup Pathak and
  7. Venkatesh Chelvam

Published 19 Nov 2020

Beilstein Arch. 2020, 2020131. doi:10.3762/bxiv.2020.131.v1

In silico approach: Anthocyanin derivatives as potential inhibitors of the COVID-19 main protease

  1. Muhammad Ikhlas Abdjan,
  2. Khusna Arif Rakhman,
  3. Sri Handayani,
  4. Chairil Anjasmara Robo Putra and
  5. Imam Siswanto

Published 15 Sep 2020

Beilstein Arch. 2020, 2020106. doi:10.3762/bxiv.2020.106.v1

Vicinal difluorination as a C=C surrogate: an analog of piperine with enhanced solubility, photostability, and acetylcholinesterase inhibitory activity

  1. Yuvixza Lizarme-Salas,
  2. Alexandra Daryl Ariawan,
  3. Ranjala Ratnayake,
  4. Hendrik Luesch,
  5. Angela Finch and
  6. Luke Hunter

Published 12 Aug 2020

Beilstein Arch. 2020, 202093. doi:10.3762/bxiv.2020.93.v1

Published 08 May 2020

Beilstein Arch. 2020, 202060. doi:10.3762/bxiv.2020.60.v1

Published 27 Apr 2020

Beilstein Arch. 2020, 202055. doi:10.3762/bxiv.2020.55.v1

Published 21 Apr 2020

Beilstein Arch. 2020, 202053. doi:10.3762/bxiv.2020.53.v1

Design, synthesis and biological evaluation of novel 5-bromo derivatives of indole phytoalexins

  1. Mariana Budovská,
  2. Ivana Selešová,
  3. Viera Tischlerová,
  4. Radka Michalková and
  5. Ján Mojžiš

Published 05 Mar 2020

Beilstein Arch. 2020, 202023. doi:10.3762/bxiv.2020.23.v1

Published 12 Feb 2020

Beilstein Arch. 2020, 202017. doi:10.3762/bxiv.2020.17.v1

Smart DNA biosensor for in vitro detection of androgen receptor mRNA

  1. Ekaterina Alexandrovna Bryushkova,
  2. Erik Rafikovich Gandalipov and
  3. Julia Victorovna Nuzhina

Published 23 Jan 2020

Beilstein Arch. 2020, 202013. doi:10.3762/bxiv.2020.13.v1

Syntheses of xanthone derivatives and their bioactivity investigation

  1. Beidou Zhou,
  2. Zhimin Weng,
  3. Yugui Tong,
  4. Zetong Ma,
  5. Rongrong Wei,
  6. Jiali Li and
  7. Zihan Yu

Published 27 Nov 2019

Beilstein Arch. 2019, 2019148. doi:10.3762/bxiv.2019.148.v1

NOVEL COMPOUNDS FROM CONDENSATION REACTION BETWEEN 2-ACETYLPYRIDINE AND 2-FORMYLPYRIDINE. SYNTHESIS, CRYSTAL STRUCTURE AND BIOLOGICAL EVALUATION

  1. Roman Vasile Rusnac,
  2. Maria Stefan Botnaru,
  3. Nicanor Barba,
  4. Peter Alexei Petrenko,
  5. Yurii Chumakov and
  6. Aurelian Petru Gulea

Published 18 Nov 2019

Beilstein Arch. 2019, 2019145. doi:10.3762/bxiv.2019.145.v1

Synthesis and cytotoxicity of novel oxindoles dispiro derivatives with thiohydantoin and adamantane fragments

  1. Maxim E. Kukushkin,
  2. Dmitriy A. Skvortsov,
  3. Marina A. Kalinina,
  4. Viktor A. Tafeenko,
  5. Vladimir V. Burmistrov,
  6. Gennady M. Butov,
  7. Nikolai V. Zyk,
  8. Alexander G. Majouga and
  9. Elena K. Beloglazkina

Published 11 Nov 2019

Beilstein Arch. 2019, 2019143. doi:10.3762/bxiv.2019.143.v1

Published 17 Oct 2019

Beilstein Arch. 2019, 2019124. doi:10.3762/bxiv.2019.124.v1

Synthesis, structural characterization and biological activity of new pyrazolo[4,3-e][1,2,4]triazine acyclonucleosides

  1. Mariusz Mojzych,
  2. Zbigniew Karczmarzyk,
  3. Joanna Matysiak and
  4. Andrzej Fruziński

Published 09 Sep 2019

Beilstein Arch. 2019, 2019102. doi:10.3762/bxiv.2019.102.v1

Published 20 Aug 2019

Beilstein Arch. 2019, 201986. doi:10.3762/bxiv.2019.86.v1

An improved, scalable synthesis of Notum inhibitor LP-922056 using 1-chloro-1,2-benziodoxol-3-one as a superior electrophilic chlorinating agent

  1. Nicky J Willis,
  2. Elliott D Bayle,
  3. George Papageorgiou,
  4. David Steadman,
  5. Benjamin N Aktinson,
  6. William Mahy and
  7. Paul V Fish

Published 16 Jul 2019

Beilstein Arch. 2019, 201970. doi:10.3762/bxiv.2019.70.v1

A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light

  1. Xavier Gómez-Santacana,
  2. Sabrina M. de Munnik,
  3. Tamara A. M. Mocking,
  4. Niels J. Hauwert,
  5. Shanliang Sun,
  6. Prashanna Vijayachandran,
  7. Iwan J. P. de Esch,
  8. Henry F. Vischer,
  9. Maikel Wijtmans and
  10. Rob Leurs

Published 15 Jul 2019

Beilstein Arch. 2019, 201969. doi:10.3762/bxiv.2019.69.v1

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