TY - JOUR
A1 - Tang, Yong-Qin
A1 - Fei, Xing-Hai
A1 - An, Jian-Xiong
A1 - Yang, Fen-Fen
A1 - Duan, Dong-Zhu
A1 - Cao, Zuo-Xian
A1 - Fu, Xiao-Zhong
A1 - Yang, Yuan-Yong
A1 - He, Bin
A1 - Zhao, Yong-Long
T1 - Palladium-catalyzed Conia-ene Reaction of 1-alkynylindolin-3-ones: a strategy for the construction of Pyrrolo[1,2-a]indoles
JF - Beilstein Archives
Y1 - 2019///
SN -
M3 - doi:10.3762/bxiv.2019.59.v1
N2 - A palladium-catalyzed conia-ene reaction of 1-alkynylindolin-3-ones has been developed. Three examples of pyrrolo[1,2-a]indoline derivatives were readily obtained with yields up to 82% utilizing this strategy. Importantly, this palladium-catalyzed intramolecular cyclization process represents an important contribution to the application of indole-3-one derivatives.
ER -