Novel Bis-Triazole Scaffold Accessed via Two Tandem [3+2] Cycloaddition Events Including an Uncatalyzed, Room-Temperature Azide-Alkyne Click Reaction

  • Ksenia Malkova,
  • Andrey Bubyrev,
  • Vasilisa Krivovicheva,
  • Dmitry Dar'in,
  • Alexander Bunev and
  • Mikhail Krasavin
Published 30 Sep 2022
Beilstein Arch. 2022, 202280. doi:10.3762/bxiv.2022.80.v1

Synthetic study toward diterpenoid aberrarone

  • Liang Shi,
  • Zhiyu Gao,
  • Yiqing Li,
  • Yuanhao Dai,
  • Yu Liu,
  • Lili Shi and
  • Hong-Dong Hao
Published 28 Sep 2022
Beilstein Arch. 2022, 202279. doi:10.3762/bxiv.2022.79.v1
Published 22 Sep 2022
Beilstein Arch. 2022, 202275. doi:10.3762/bxiv.2022.75.v1
Published 19 Sep 2022
Beilstein Arch. 2022, 202273. doi:10.3762/bxiv.2022.73.v1

Rhodium-catalyzed intramolecular reductive aldol-type cyclization: Application for the synthesis of a chiral necic acid lactone

  • Motoyuki Isoda,
  • Kazuyuki Sato,
  • Kenta Kameda,
  • Kana Wakabayashi,
  • Ryota Sato,
  • Hideki Minami,
  • Yukiko Karuo,
  • Atsushi Tarui,
  • Kentaro Kawai and
  • Masaaki Omote
Published 16 Sep 2022
Beilstein Arch. 2022, 202272. doi:10.3762/bxiv.2022.72.v1

One-pot Double Annulations to Confer Diastereoselective Spirooxindole-pyrrolothiazoles

  • Juan Lu,
  • Bin Yao,
  • Desheng Zhan,
  • Zhuo Sun,
  • Yun Ji and
  • Xiaofeng Zhang
Published 14 Sep 2022
Beilstein Arch. 2022, 202271. doi:10.3762/bxiv.2022.71.v1

Formal Total Synthesis of Macarpine via a Au(I)-Catalyzed 6-endo-dig Cycloisomerization Strategy

  • Jiayue Fu,
  • Bingbing Li,
  • Zefang Zhou,
  • Maosheng Cheng,
  • Lu Yang and
  • Yongxiang Liu
Published 14 Sep 2022
Beilstein Arch. 2022, 202270. doi:10.3762/bxiv.2022.70.v1
Published 23 Aug 2022
Beilstein Arch. 2022, 202269. doi:10.3762/bxiv.2022.69.v1

Comparison of crystal structure and DFT calculation of triferrocenyl trithiophosphite’s conformation

  • Ruslan P. Shekurov,
  • Mikhail N. Khrizanforov,
  • Ilya A. Bezkishko,
  • Tatiana P. Gerasimova,
  • Almaz A. Zagidullin,
  • Daut R. Islamov and
  • Vasili A. Miluykov
Published 18 Aug 2022
Beilstein Arch. 2022, 202268. doi:10.3762/bxiv.2022.68.v1

ULTRASOUND-ASSISTED GREEN SYNTHESES OF NOVEL PYRIMIDINE DERIVATIVES AND THEIR COMPARISON WITH CONVENTIONAL METHODS

  • Vergush A. Pivazyan,
  • Emma A. Ghazaryan,
  • Armen V. Karapetyan,
  • Roza S. Shainova,
  • Siranush V. Harutyunyan,
  • Asya S. Vorskanyan,
  • Aleksandr P. Yengoyan and
  • Tiruhi A. Gomktsyan
Published 16 Aug 2022
Beilstein Arch. 2022, 202267. doi:10.3762/bxiv.2022.67.v1

Synthesis of 3,4,5-tris(chlorophenyl)-1,2-diphosphaferrocenes and their electrochemical properties

  • Almaz A. Zagidullin,
  • Farida Akhmatkhanova,
  • Mikhail Khrizanforov,
  • Robert Fayzullin,
  • Tatiana Gerasimova,
  • Ilya A. Bezkishko and
  • Vasili Miluykov
Published 11 Jul 2022
Beilstein Arch. 2022, 202261. doi:10.3762/bxiv.2022.61.v1
Published 05 Jul 2022
Beilstein Arch. 2022, 202259. doi:10.3762/bxiv.2022.59.v1

Synthesis of Protected Precursors of Chitin Oligosaccharides by Electrochemical Polyglycosylation of Thioglycosides

  • Md Azadur Rahman,
  • Kana Kuroda,
  • Hirofumi Endo,
  • Norihiko Sasaki,
  • Tomoaki Hamada,
  • Hiraku Sakai and
  • Toshiki Nokami
Published 04 Jul 2022
Beilstein Arch. 2022, 202258. doi:10.3762/bxiv.2022.58.v1

Synthesis of C6-modified mannose 1-phosphates and evaluation of derived sugar nucleotides against GDP‑mannose dehydrogenase

  • Sanaz Ahmadipour,
  • Alice J C Wahart,
  • Jonathan P Dolan,
  • Laura Beswick,
  • Chris S Hawes,
  • Robert A Field and
  • Gavin J Miller
Published 04 Jul 2022
Beilstein Arch. 2022, 202257. doi:10.3762/bxiv.2022.57.v1

Heterogeneous metallaphotoredox catalysis in a continuous-flow packed bed reactor

  • Wei-Hsin Hsu,
  • Susanne Reischauer,
  • Peter H Seeberger,
  • Bartholomäus Pieber and
  • Dario Cambié
Published 29 Jun 2022
Beilstein Arch. 2022, 202256. doi:10.3762/bxiv.2022.56.v1
Published 22 Jun 2022
Beilstein Arch. 2022, 202253. doi:10.3762/bxiv.2022.53.v1

Facile and Diastereoselective Arylation of the Privileged 1,4-Dihydroisoquinolin-3(2H)-one Scaffold

  • Dmitry Dar'in,
  • Grigory Kantin,
  • Alexander Bunev and
  • Mikhail Krasavin
Published 20 Jun 2022
Beilstein Arch. 2022, 202250. doi:10.3762/bxiv.2022.50.v1
Published 13 Jun 2022
Beilstein Arch. 2022, 202249. doi:10.3762/bxiv.2022.49.v1

Characterization of a new fusicoccane-type diterpene synthase and an associated P450 enzyme

  • Jia-Hua Huang,
  • Jian-Ming Lv,
  • Liang-Yan Xiao,
  • Qian Xu,
  • Fu-long Lin,
  • Gao-Qian Wang,
  • Guo-Dong Chen,
  • Sheng-Ying Qin,
  • Dan Hu and
  • Hao Gao
Published 09 Jun 2022
Beilstein Arch. 2022, 202247. doi:10.3762/bxiv.2022.47.v1

Mechanochemical bottom-up synthesis of phosphorus-linked, heptazine-based carbon nitrides using sodium phosphide

  • Blaine G. Fiss,
  • Georgia Douglas,
  • Michael Ferguson,
  • Jorge Becerra,
  • Jesus Valdez,
  • Trong-On Do,
  • Tomislav Friscic and
  • Audrey H. Moores
Published 07 Jun 2022
Beilstein Arch. 2022, 202245. doi:10.3762/bxiv.2022.45.v1
Published 07 Jun 2022
Beilstein Arch. 2022, 202244. doi:10.3762/bxiv.2022.44.v1
Published 03 Jun 2022
Beilstein Arch. 2022, 202243. doi:10.3762/bxiv.2022.43.v1
Published 31 May 2022
Beilstein Arch. 2022, 202240. doi:10.3762/bxiv.2022.40.v1
Published 30 May 2022
Beilstein Arch. 2022, 202239. doi:10.3762/bxiv.2022.39.v1
Published 27 May 2022
Beilstein Arch. 2022, 202238. doi:10.3762/bxiv.2022.38.v1
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